SCHEMBL4046819

SCHEMBL4046819

CC(C(c1ccc(-c2ccc(C(C)(C)O)nn2)cc1)(c1ccc(OCc2ncccn2)cn1)S(C)(=O)=O)S(C)(=O)=O

nearest known ligand 0.53

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALOX5AP P20292 3/20 0.53
CYP4F2 P78329 4/20 0.33
CYP4A11 Q02928 4/20 0.33
ADAMTS4 O75173 4/20 0.32
MAPT P10636 1/20 0.31
PDE10A Q9Y233 1/20 0.31
MMP13 P45452 2/20 0.31
PPARD Q03181 1/20 0.30
DGAT1 O75907 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL706833 0.82 ALOX5AP (0.72) ALOX5APCYP4F2CYP4A11ADAMTS4PDE10A
SCHEMBL706834 0.82 ALOX5AP (0.72) ALOX5APCYP4F2CYP4A11ADAMTS4PDE10A
SCHEMBL708386 0.73 ALOX5AP (0.90) ALOX5APCYP4F2CYP4A11ADAMTS4MAPT
SCHEMBL708385 0.73 ALOX5AP (0.90) ALOX5APCYP4F2CYP4A11ADAMTS4MAPT
SCHEMBL710361 0.72 ALOX5AP (0.58) ALOX5APCYP4F2CYP4A11ADAMTS4MMP13
SCHEMBL480273 0.69 ALOX5AP (1.00) ALOX5APADAMTS4MAPT
SCHEMBL707622 0.69 ALOX5AP (0.63) ALOX5APCYP4F2CYP4A11PDE10AMMP13
SCHEMBL709308 0.69 ALOX5AP (0.63) ALOX5APCYP4F2CYP4A11PDE10AMMP13
SCHEMBL2997218 0.68 ALOX5AP (0.55) ALOX5APADAMTS4MAPTMMP13PPARD
SCHEMBL2997435 0.68 ALOX5AP (0.86) ALOX5APADAMTS4MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2013174-A2 DIARYL SUBSTITUTED ALKANES Merck & Co., Inc. (US) 2009-01-14 EP disclosed
WO-2007120574-A2 DIARYL SUBSTITUTED ALKANES MERCK & CO., INC. (US) 2007-10-25 WO disclosed