SCHEMBL4048743

SCHEMBL4048743

CC(C)(C)[C@H](NC(=O)c1nn(CC2CCOCC2)c2cc(F)ccc12)C(=O)NCCNS(=O)(=O)C1CC1

nearest known ligand 0.44

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 6/20 0.44
CNR1 P21554 7/20 0.38
GRM4 Q14833 4/20 0.36
CNR2 P34972 6/20 0.36
ROCK2 O75116 1/20 0.35
HTR3A P46098 1/20 0.34
HTR4 Q13639 2/20 0.34
CYP3A4 P08684 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13691018 1.00 ROCK1 (0.44) ROCK1CNR1GRM4CNR2ROCK2
SCHEMBL13690641 0.90 ROCK1 (0.47) ROCK1CNR1GRM4CNR2ROCK2
SCHEMBL4053793 0.90 ROCK1 (0.47) ROCK1CNR1GRM4CNR2ROCK2
SCHEMBL13691270 0.89 ROCK1 (0.46) ROCK1CNR1GRM4CNR2ROCK2
SCHEMBL13690669 0.87 ROCK1 (0.44) ROCK1CNR1GRM4CNR2HTR3A
SCHEMBL4056281 0.86 ROCK1 (0.43) ROCK1CNR1GRM4CNR2HTR4
SCHEMBL4056397 0.86 CNR1 (0.37) ROCK1CNR1GRM4CNR2ROCK2
SCHEMBL13690608 0.85 ROCK1 (0.43) ROCK1CNR1GRM4CNR2HTR3A
SCHEMBL13691036 0.85 CNR1 (0.42) ROCK1CNR1CNR2HTR3A
SCHEMBL4050830 0.85 ROCK1 (0.44) ROCK1CNR1GRM4CNR2HTR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009106980-A2 INDAZOLE DERIVATIVES PFIZER INC. (US) 2009-09-03 WO claimed