SCHEMBL13690641

SCHEMBL13690641

CC(C)(C)C(NC(=O)c1nn(CC2CCOCC2)c2cc(F)ccc12)C(=O)NCCO

nearest known ligand 0.47

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 6/20 0.47
CNR1 P21554 6/20 0.40
GRM4 Q14833 4/20 0.38
CNR2 P34972 5/20 0.38
HTR3A P46098 1/20 0.36
HTR4 Q13639 3/20 0.36
CYP3A4 P08684 1/20 0.36
ROCK2 O75116 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4053793 1.00 ROCK1 (0.47) ROCK1CNR1GRM4CNR2HTR3A
SCHEMBL13691270 0.95 ROCK1 (0.46) ROCK1CNR1GRM4CNR2HTR3A
SCHEMBL13690964 0.94 ROCK1 (0.47) ROCK1CNR1GRM4CNR2HTR3A
SCHEMBL4057153 0.94 ROCK1 (0.47) ROCK1CNR1GRM4CNR2HTR3A
SCHEMBL4052498 0.92 CNR1 (0.49) ROCK1CNR1CNR2HTR3AHTR4
SCHEMBL13691275 0.92 CNR1 (0.49) ROCK1CNR1CNR2HTR3AHTR4
SCHEMBL13690669 0.90 ROCK1 (0.44) ROCK1CNR1GRM4CNR2HTR3A
SCHEMBL4048743 0.90 ROCK1 (0.44) ROCK1CNR1GRM4CNR2HTR3A
SCHEMBL13691018 0.90 ROCK1 (0.44) ROCK1CNR1GRM4CNR2HTR3A
SCHEMBL4050830 0.90 ROCK1 (0.44) ROCK1CNR1GRM4CNR2HTR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009106980-A2 INDAZOLE DERIVATIVES PFIZER INC. (US) 2009-09-03 WO disclosed