SCHEMBL4052185

SCHEMBL4052185

CN1Cc2c(N3CCOCC3)nc3sc4c(=O)[nH]cnc4c3c2CC1(C)C

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.73
ALDH1A1 P00352 5/20 0.73
HPGD P15428 2/20 0.73
HIF1A Q16665 2/20 0.73
PDE4B Q07343 7/20 0.61
HSD17B10 Q99714 2/20 0.56
TSHR P16473 1/20 0.56
MAPK1 P28482 2/20 0.54
MAPT P10636 3/20 0.53
NPSR1 Q6W5P4 3/20 0.53
RAD52 P43351 1/20 0.53
ATM Q13315 1/20 0.53
APAF1 O14727 1/20 0.51
GPR55 Q9Y2T6 1/20 0.51
HKDC1 Q2TB90 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
PDE4A P27815 3/20 0.47
PDE4D Q08499 3/20 0.47
LMNA P02545 1/20 0.47
AGTR1 P30556 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL424777 0.86 ALDH1A1 (0.74) KDM4EALDH1A1HPGDHIF1APDE4B
SCHEMBL4044859 0.84 ALDH1A1 (0.74) KDM4EALDH1A1HPGDHIF1APDE4B
SCHEMBL4049404 0.81 PDE4B (0.70) KDM4EALDH1A1HPGDPDE4BHSD17B10
SCHEMBL432053 0.81 ALDH1A1 (0.70) KDM4EALDH1A1HPGDHIF1APDE4B
SCHEMBL427971 0.81 ALDH1A1 (0.68) KDM4EALDH1A1HPGDHIF1AHSD17B10
SCHEMBL4053824 0.80 ALDH1A1 (0.67) KDM4EALDH1A1HPGDHIF1APDE4B
SCHEMBL5015896 0.79 ALDH1A1 (0.61) KDM4EALDH1A1HPGDHIF1APDE4B
SCHEMBL4045742 0.79 KDM4E (0.66) KDM4EALDH1A1HPGDHIF1APDE4B
SCHEMBL5011421 0.79 ALDH1A1 (0.67) KDM4EALDH1A1HPGDHIF1APDE4B
SCHEMBL5015893 0.78 ALDH1A1 (0.66) KDM4EALDH1A1HPGDHIF1APDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1819710-B1 NEW PYRIDOTHIENOPYRIMIDINE DERIVATIVES ALMIRALL LAB (ES) 2009-03-11 EP disclosed