SCHEMBL4052797

SCHEMBL4052797

COc1ccc(C2(C#N)CCc3ncncc3C2)c2c1oc1ccc(NS(C)(=O)=O)cc12

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PDE4D Q08499 1/20 0.38
CYP17A1 P05093 9/20 0.37
PDE4B Q07343 2/20 0.33
KIT P10721 2/20 0.32
USP2 O75604 2/20 0.32
ALDH1A1 P00352 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
KDM1A O60341 1/20 0.31
RET P07949 1/20 0.31
LRRK2 Q5S007 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C19 P33261 1/20 0.31
HSD17B10 Q99714 1/20 0.31
CLK4 Q9HAZ1 1/20 0.31
IDO1 P14902 1/20 0.31
TDO2 P48775 1/20 0.31
TP53 P04637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4051940 0.91 PDE4D (0.48) PDE4DCYP17A1PDE4B
SCHEMBL4062007 0.85 HRH4 (0.31)
SCHEMBL4018297 0.84 CYP17A1 (0.33) CYP17A1PDE4BALDH1A1HSD17B10
SCHEMBL4053327 0.84 CYP17A1 (0.37) CYP17A1KITUSP2KDM1ACYP1A2
SCHEMBL4059118 0.81 CYP17A1 (0.35) PDE4DCYP17A1PDE4B
SCHEMBL4060696 0.76 HRH4 (0.37)
SCHEMBL4013156 0.74 HRH4 (0.33) CYP17A1PDE4BALDH1A1
SCHEMBL4235894 0.73 HRH4 (0.35)
SCHEMBL14865178 0.73 PDE4B (0.33) CYP17A1PDE4BALDH1A1
SCHEMBL4059123 0.72

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009115874-A2 NOVEL HETEROCYCLIC COMPOUNDS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCESSES FOR THEIR PREPARATION MATRIX LABORATORIES LTD. (IN) 2009-09-24 WO claimed
WO-2009115874-A2 NOVEL HETEROCYCLIC COMPOUNDS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCESSES FOR THEIR PREPARATION MATRIX LABORATORIES LTD. (IN) 2009-09-24 WO disclosed