SCHEMBL4053887

SCHEMBL4053887

CNCCCN1c2cccc(C)c2N(c2ccccc2)S1(O)O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 20/20 0.46
SLC6A4 P31645 7/20 0.46
SLC6A3 Q01959 5/20 0.42
KCNH2 Q12809 2/20 0.37
CYP3A4 P08684 2/20 0.37
SLC22A2 O15244 1/20 0.37
SLC22A1 O15245 1/20 0.37
SLC22A3 O75751 1/20 0.37
CYP1A2 P05177 1/20 0.37
CHRM2 P08172 1/20 0.37
CYP2D6 P10635 1/20 0.37
CHRM1 P11229 1/20 0.37
DRD2 P14416 1/20 0.37
ADRA2B P18089 1/20 0.37
ADRA2C P18825 1/20 0.37
NFKB1 P19838 1/20 0.37
CHRM3 P20309 1/20 0.37
HTR2A P28223 1/20 0.37
HTR2C P28335 1/20 0.37
MAPK1 P28482 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4054031 0.87 SLC6A2 (0.52) SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL4053883 0.85 SLC6A2 (0.56) SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL4059292 0.84 SLC6A2 (0.53) SLC6A2SLC6A4SLC6A3KCNH2CYP3A4
SCHEMBL4053619 0.81 SLC6A2 (0.52) SLC6A2SLC6A4SLC6A3KCNH2CYP3A4
SCHEMBL4053529 0.81 SLC6A2 (0.54) SLC6A2SLC6A4SLC6A3KCNH2CYP3A4
Hydrochloric Acid SCHEMBL4947362 0.80 SLC6A2 (0.53) SLC6A2SLC6A4SLC6A3KCNH2CYP3A4
SCHEMBL4055129 0.80 SLC6A2 (0.52) SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL4059522 0.79 SLC6A2 (0.54) SLC6A2SLC6A4SLC6A3KCNH2CYP3A4
SCHEMBL4947338 0.78 SLC6A2 (0.43) SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL4052761 0.78 SLC6A2 (0.43) SLC6A2SLC6A4SLC6A3KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2061776-A1 ARYL SULFAMIDE DERIVATIVES AND METHODS OF THEIR USE Wyeth a Corporation of the State of Delaware (US) 2009-05-27 EP claimed
WO-2008073459-A1 ARYL SULFAMIDE DERIVATIVES AND METHODS OF THEIR USE WYETH (US) 2008-06-19 WO claimed
EP-2061776-A1 ARYL SULFAMIDE DERIVATIVES AND METHODS OF THEIR USE Wyeth a Corporation of the State of Delaware (US) 2009-05-27 EP disclosed
WO-2008073459-A1 ARYL SULFAMIDE DERIVATIVES AND METHODS OF THEIR USE WYETH (US) 2008-06-19 WO disclosed