SCHEMBL4054063

SCHEMBL4054063

CC(C)(C)OC(=O)NCc1ccc(Cn2nnc3c(-c4ccco4)nc(N)nc32)cc1.Nc1nc(-c2ccco2)c2nnn(Cc3cccc4[nH]ccc34)c2n1

nearest known ligand 0.56

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 20/20 0.56
ADORA2B P29275 20/20 0.56
ADORA1 P30542 20/20 0.56
ADORA3 P0DMS8 19/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4048625 0.90 ADORA2A (0.67) ADORA2AADORA2BADORA1ADORA3
SCHEMBL4047229 0.85 ADORA3 (0.64) ADORA2AADORA2BADORA1ADORA3
SCHEMBL4225098 0.85 ADORA2A (0.69) ADORA2AADORA2BADORA1ADORA3
SCHEMBL4045905 0.83 ADORA2A (0.71) ADORA2AADORA2BADORA1ADORA3
SCHEMBL4054064 0.82 ADORA2A (0.52) ADORA2AADORA2BADORA1ADORA3
SCHEMBL4048192 0.81 ADORA2A (0.59) ADORA2AADORA2BADORA1ADORA3
SCHEMBL4045607 0.78 ADORA2A (0.76) ADORA2AADORA2BADORA1ADORA3
SCHEMBL4049496 0.77 ADORA2A (0.64) ADORA2AADORA2BADORA1ADORA3
SCHEMBL4046235 0.77 ADORA3 (0.57) ADORA2AADORA2BADORA1ADORA3
SCHEMBL4043357 0.76 ADORA3 (0.59) ADORA2AADORA2BADORA1ADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1392312-B1 TRIAZOLO 4,5-d PYRIMIDINE DERIVATIVES AND THEIR USE AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RES LTD (GB) 2009-03-04 EP claimed