SCHEMBL4054776

SCHEMBL4054776

Cc1cc(Cn2nnc3c(-c4ccco4)nc(N)nc32)c2c(ccn2C(=O)O)c1

nearest known ligand 0.62

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 20/20 0.62
ADORA2A P29274 20/20 0.62
ADORA2B P29275 20/20 0.62
ADORA1 P30542 20/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4048337 0.91 ADORA2A (0.62) ADORA3ADORA2AADORA2BADORA1
SCHEMBL4051302 0.90 ADORA3 (0.56) ADORA3ADORA2AADORA2BADORA1
SCHEMBL4049592 0.89 ADORA2A (0.65) ADORA3ADORA2AADORA2BADORA1
SCHEMBL4051305 0.84 ADORA3 (0.58) ADORA3ADORA2AADORA2BADORA1
SCHEMBL4045523 0.82 ADORA3 (0.55) ADORA3ADORA2AADORA2BADORA1
SCHEMBL4045081 0.81 ADORA2A (0.69) ADORA3ADORA2AADORA2BADORA1
SCHEMBL4043444 0.81 ADORA2A (0.64) ADORA3ADORA2AADORA2BADORA1
SCHEMBL4046852 0.81 ADORA2A (0.69) ADORA3ADORA2AADORA2BADORA1
SCHEMBL4045557 0.81 ADORA2A (0.76) ADORA3ADORA2AADORA2BADORA1
SCHEMBL4045750 0.80 ADORA3 (0.53) ADORA3ADORA2AADORA2BADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1392312-B1 TRIAZOLO 4,5-d PYRIMIDINE DERIVATIVES AND THEIR USE AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RES LTD (GB) 2009-03-04 EP claimed