SCHEMBL4054846

SCHEMBL4054846

COc1ccc2nccc(N3CCC(C(N)CN)C3I)c2n1

nearest known ligand 0.39

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 7/20 0.36
CYP8B1 Q9UNU6 1/20 0.35
SLC2A1 P11166 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3178305 0.78 CYP8B1 (0.44) KCNH2CYP8B1
SCHEMBL3179377 0.71 CYP8B1 (0.46) KCNH2CYP8B1
SCHEMBL1224385 0.71 CYP8B1 (0.46) KCNH2CYP8B1
SCHEMBL3665601 0.71 CYP8B1 (0.46) KCNH2CYP8B1
SCHEMBL4066839 0.71 CYP8B1 (0.46) KCNH2CYP8B1
SCHEMBL1222834 0.71 CYP2C19 (0.46) KCNH2CYP8B1
SCHEMBL10078632 0.70 HTR2C (0.45) KCNH2CYP8B1
SCHEMBL1222886 0.70 CYP8B1 (0.41) KCNH2CYP8B1
SCHEMBL3636416 0.69 CYP2C19 (0.54) KCNH2CYP8B1
SCHEMBL3634872 0.69 CYP2C19 (0.54) KCNH2CYP8B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1773343-A4 ANTIBACTERIAL AGENTS GLAXO GROUP LTD (GB) 2009-05-13 EP disclosed
EP-1773343-A1 ANTIBACTERIAL AGENTS GLAXO GROUP LIMITED (GB) 2007-04-18 EP disclosed
WO-2006017326-A1 ANTIBACTERIAL AGENTS GLAXO GROUP LIMITED (GB) 2006-02-16 WO disclosed