SCHEMBL4057735

SCHEMBL4057735

CCCC(O)(/C(=C\I)C(=O)O)c1ccccc1C

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 3/20 0.35
CYP2C19 P33261 3/20 0.35
ALOX12 P18054 1/20 0.35
CTBP2 P56545 1/20 0.34
ALDH1A1 P00352 3/20 0.33
KDM4E B2RXH2 2/20 0.33
NPSR1 Q6W5P4 2/20 0.33
ATM Q13315 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
EGFR P00533 1/20 0.33
MMP1 P03956 1/20 0.33
MMP2 P08253 1/20 0.33
MMP9 P14780 1/20 0.33
ERCC5 P28715 1/20 0.33
FEN1 P39748 1/20 0.33
CHRM3 P20309 2/20 0.32
CHRM2 P08172 1/20 0.32
CHRM1 P11229 1/20 0.32
LMNA P02545 3/20 0.32
CYP1A2 P05177 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4057738 1.00 GAA (0.35) GAACYP2C19ALOX12CTBP2ALDH1A1
SCHEMBL4060400 0.83 CYP2C19 (0.40) GAACYP2C19ALOX12ALDH1A1KDM4E
SCHEMBL4060403 0.83 CYP2C19 (0.40) GAACYP2C19ALOX12ALDH1A1KDM4E
SCHEMBL4058650 0.72 CYP3A4 (0.39) CYP2C19NPSR1CYP1A2CYP3A4CYP2D6
SCHEMBL4058658 0.72 CYP3A4 (0.39) CYP2C19NPSR1CYP1A2CYP3A4CYP2D6
SCHEMBL3504696 0.72 HPGD (0.38) GAACTBP2ALDH1A1KDM4ENPSR1
SCHEMBL4059130 0.70 ALDH1A1 (0.45) ALDH1A1KDM4EATMTDP1MMP9
SCHEMBL28892811 0.70 CYP2C19 (0.39) GAACYP2C19ALOX12CTBP2ALDH1A1
SCHEMBL20210869 0.69 CASR (0.39) GAACYP2C19ALOX12ATMCHRM3
SCHEMBL4057733 0.69 GAA (0.43) GAACYP2C19ALDH1A1KDM4EATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009110655-A1 NOVEL BETA SUBSTITUTED MORITA-BAYLIS-HILLMAN DERIVATIVES SUNGKYUNKWAN UNIVERSITY FOUNDATION FOR CORPORATE COLLABORATION (KR) 2009-09-11 WO disclosed