SCHEMBL4058224

SCHEMBL4058224

CC(=O)[C@@](O)(C(N)=O)[C@@H](O)[C@H](O)[C@H](O)CO

nearest known ligand 0.37

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
USP2 O75604 1/20 0.37
SLCO1B1 Q9Y6L6 1/20 0.37
LMNA P02545 2/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
PDE4A P27815 1/20 0.35
TDP1 Q9NUW8 1/20 0.34
KDM4E B2RXH2 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2000595 1.00 USP2 (0.37) USP2SLCO1B1LMNAL3MBTL1PDE4A
SCHEMBL2789359 1.00 USP2 (0.37) USP2SLCO1B1LMNAL3MBTL1PDE4A
SCHEMBL27550874 1.00 USP2 (0.37) USP2SLCO1B1LMNAL3MBTL1PDE4A
SCHEMBL5859311 0.83 PDE4A (0.41) USP2SLCO1B1LMNAL3MBTL1PDE4A
SCHEMBL16798768 0.83 PDE4A (0.41) USP2SLCO1B1LMNAL3MBTL1PDE4A
SCHEMBL29162767 0.83 PDE4A (0.41) USP2SLCO1B1LMNAL3MBTL1PDE4A
SCHEMBL29020598 0.82 LMNA (0.46) USP2SLCO1B1LMNAL3MBTL1PDE4A
SCHEMBL19717486 0.82
SCHEMBL17260872 0.82 USP2 (0.35) USP2SLCO1B1LMNAL3MBTL1PDE4A
SCHEMBL941684 0.81 LMNA (0.36) USP2SLCO1B1LMNAL3MBTL1PDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3423457-A1 PROCESS FOR THE PREPARATION OF AN ANTIBODY-RIFAMYCIN CONJUGATE H. Hoffnabb-La Roche Ag (CH) 2019-01-09 EP disclosed
EP-3226911-A1 ANTI-STAPHYLOCOCCUS AUREUS ANTIBODY RIFAMYCIN CONJUGATES AND USES THEREOF F.HOFFMANN-LA ROCHE AG (CH) 2017-10-11 EP disclosed
WO-2016090038-A1 ANTI-STAPHYLOCOCCUS AUREUS ANTIBODY RIFAMYCIN CONJUGATES AND USES THEREOF GENENTECH, INC. (US) 2016-06-09 WO disclosed
EP-3004162-A1 ANTI-WALL TEICHOIC ANTIBODIES AND CONJUGATES Genentech, Inc. (US) 2016-04-13 EP disclosed
EP-3004161-A1 ANTI-WALL TEICHOIC ANTIBODIES AND CONJUGATES Genentech, Inc. (US) 2016-04-13 EP disclosed
WO-2014194247-A1 ANTI-WALL TEICHOIC ANTIBODIES AND CONJUGATES GENENTECH, INC. (US) 2014-12-04 WO disclosed
WO-2014193722-A1 ANTI-WALL TEICHOIC ANTIBODIES AND CONJUGATES GENENTECH, INC. (US) 2014-12-04 WO disclosed
US-7528113-B2 Method and composition for the treatment of adenoviral ocular infections ADENOVIR PHARMA AB (SE) 2009-05-05 US disclosed
EP-1231925-B1 METHOD AND COMPOSITION FOR THE TREATMENT OF ADENOVIRAL OCULAR INFECTIONS WADELL GOERAN (SE) 2005-06-08 EP disclosed
US-20050080041-A1 Method and composition for the treatment of adenoviral ocular infections ADENOVIR PHARMA AB (SE) 2005-04-14 US disclosed
EP-1231925-A1 METHOD AND COMPOSITION FOR THE TREATMENT OF ADENOVIRAL OCULAR INFECTIONS Wadell, Göran (SE) 2002-08-21 EP disclosed
WO-2001037846-A1 METHOD AND COMPOSITION FOR THE TREATMENT OF ADENOVIRAL OCULAR INFECTIONS WADELL GOERAN (SE) 2001-05-31 WO disclosed