Diphenyl Borinic Acid

Diphenyl Borinic Acid

SCHEMBL40601

OB(c1ccccc1)c1ccccc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV6 Q9H1D0 7/20 1.00
ORAI1 Q96D31 6/20 1.00
ORAI2 Q96SN7 6/20 1.00
ORAI3 Q9BRQ5 6/20 1.00
PCSK9 Q8NBP7 2/20 1.00
CA4 P22748 2/20 0.65
CA14 Q9ULX7 2/20 0.65
ENPP2 Q13822 2/20 0.65
CA6 P23280 1/20 0.65
CA5A P35218 1/20 0.65
CA7 P43166 1/20 0.65
CA5B Q9Y2D0 1/20 0.65
MGLL Q99685 2/20 0.46
CA1 P00915 5/20 0.46
CA2 P00918 4/20 0.46
CA12 O43570 1/20 0.39
GLA P06280 1/20 0.39
CA3 P07451 1/20 0.39
CA9 Q16790 1/20 0.39
TDP1 Q9NUW8 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Diphenyl Borinic Acid SCHEMBL28080639 0.97 TRPV6 (0.93) TRPV6ORAI1ORAI2ORAI3PCSK9
SCHEMBL2412647 0.97 TRPV6 (0.93) TRPV6ORAI1ORAI2ORAI3PCSK9
SCHEMBL2406379 0.91 TRPV6 (0.82) TRPV6ORAI1ORAI2ORAI3PCSK9
SCHEMBL2406124 0.88 TRPV6 (0.78) TRPV6ORAI1ORAI2ORAI3PCSK9
Diphenyl Borinic Acid SCHEMBL20694919 0.88 TRPV6 (0.78) TRPV6ORAI1ORAI2ORAI3PCSK9
SCHEMBL2407457 0.86 TRPV6 (0.74) TRPV6ORAI1ORAI2ORAI3PCSK9
SCHEMBL2405808 0.84 TRPV6 (0.72) TRPV6ORAI1ORAI2ORAI3PCSK9
SCHEMBL17698481 0.84 TRPV6 (0.70) TRPV6ORAI1ORAI2ORAI3PCSK9
SCHEMBL3275714 0.84 TRPV6 (0.70) TRPV6ORAI1ORAI2ORAI3PCSK9
SCHEMBL12266144 0.84 TRPV6 (0.80) TRPV6ORAI1ORAI2ORAI3PCSK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 3985 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3662012-B1 HANDLING ADDITIVE FOR SILICONE ELASTOMER BASES DOW SILICONES CORP (US) 2024-08-28 EP claimed
EP-3715346-B1 THIAZOLYL-CONTAINING COMPOUNDS FOR TREATING PROLIFERATIVE DISEASES DANA FARBER CANCER INST INC (US) 2024-01-03 EP claimed
EP-3606528-B1 TRICYCLIC COMPOUNDS AS GLYCOGEN SYNTHASE KINASE 3 (GSK3) INHIBITORS AND USES THEREOF BROAD INST INC (US) 2023-10-18 EP claimed
EP-4093805-A1 POLYMERS BASED ON IONIC MONOMERS, COMPOSITIONS COMPRISING SAME, METHODS FOR MANUFACTURING SAME, AND USE THEREOF IN ELECTROCHEMICAL APPLICATIONS Hydro-Québec (CA) 2022-11-30 EP claimed
US-11505676-B2 Handling additive for silicone elastomer bases DOW SILICONES CORPORATION (US) 2022-11-22 US claimed
US-11241435-B2 Uses of salt-inducible kinase (SIK) inhibitors for treating osteoporosis THE GENERAL HOSPITAL CORPORATION (US) 2022-02-08 US claimed
EP-3500551-B1 PROCESS FOR PREPARING SUBSTITUTED BIPHENYLS BASF SE (DE) 2021-11-10 EP claimed
EP-3172213-B1 MACROCYCLIC KINASE INHIBITORS AND USES THEREOF DANA FARBER CANCER INST INC (US) 2021-09-22 EP claimed
WO-2021146815-A1 POLYMERS BASED ON IONIC MONOMERS, COMPOSITIONS COMPRISING SAME, METHODS FOR MANUFACTURING SAME, AND USE THEREOF IN ELECTROCHEMICAL APPLICATIONS HYDRO-QUéBEC (CA) 2021-07-29 WO claimed
EP-3583093-B1 PROCESS FOR PREPARING SUBSTITUTED BIPHENYLS BASF SE (DE) 2021-04-14 EP claimed
WO-2003059916-A2 METHODS FOR THE PREPARATION OF ALKYL DIARYL BORINATES AND COMPLEXED DIARYLBORINIC ACIDS THE PENNSYLVANIA STATE RESEARCH FOUNDATION (US) 2003-07-24 WO claimed
EP-1140947-B1 METHOD FOR PRODUCING MONO-ORGANOBORANES OR DI-ORGANOBORANES BASELL POLYOLEFINE GMBH (DE) 2003-03-12 EP claimed
WO-2002044184-A2 DNA METHYL TRANSFERASE INHIBITORS THE PENN STATE RESEARCH FOUNDATION (US) 2002-06-06 WO claimed
EP-0881924-A1 WASTE STREAM TREATMENT E.I. DU PONT DE NEMOURS AND COMPANY (US) 1998-12-09 EP claimed
WO-1997030759-A1 WASTE STREAM TREATMENT E.I. DU PONT DE NEMOURS AND COMPANY (US) 1997-08-28 WO claimed
WO-1995005081-A1 BIOCIDAL COMPOSITIONS CONTAINING ORGANOBORON COMPOUNDS U.S. BORAX INC. (US) 1995-02-23 WO claimed
US-4931573-A CATALYTIC HYDROGENATION OF DICARBOXYLIC ACID, ESTER OR ANHYDRIDE WITH RUTHENIUM, PHOSPHINES AND GROUPS 3,4,5 COMPOUNDS MITSUBISHI KASEI CORPORATION (JP) 1990-06-05 US claimed
US-4713346-A Formation of analyzable boron containing adducts THE CHILDREN'S MEDICAL CENTER CORPORATION (US) 1987-12-15 US claimed
EP-0136683-A2 Fluorochlorohydrocarbon compositions DAIKIN INDUSTRIES, LTD. (JP) 1985-04-10 EP claimed
US-4177215-A Recovery of triarylboranes E. I. DU PONT DE NEMOURS AND COMPANY (US) 1979-12-04 US claimed