SCHEMBL4060101

SCHEMBL4060101

COC(=O)C1CNCC(C(=O)OC)C1=O

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 4/20 0.48
CHRNA4 P43681 4/20 0.48
CHRNB4 P30926 2/20 0.48
CHRNA3 P32297 2/20 0.48
CHRNA7 P36544 1/20 0.48
CYP1A2 P05177 1/20 0.38
HIF1A Q16665 1/20 0.38
BRD4 O60885 1/20 0.36
KMT2A Q03164 1/20 0.36
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13882832 0.79 CYP1A2 (0.46) CHRNB2CHRNA4CHRNB4CHRNA3CHRNA7
SCHEMBL28345166 0.76 CHRNB2 (0.39) CHRNB2CHRNA4CHRNB4CHRNA3CHRNA7
SCHEMBL567797 0.76 CHRNB2 (0.39) CHRNB2CHRNA4CHRNB4CHRNA3CHRNA7
SCHEMBL3974812 0.76 CYP1A2 (0.43) CYP1A2HIF1ABRD4ALDH1A1
Hydrochloric Acid SCHEMBL653032 0.75 CHRNB2 (0.38) CHRNB2CHRNA4CHRNB4CHRNA3CHRNA7
Hydrochloric Acid SCHEMBL22999868 0.74 CHRNB2 (0.37) CHRNB2CHRNA4CHRNB4CHRNA3CHRNA7
SCHEMBL22069021 0.74 CYP1A2 (0.36) CHRNB2CHRNA4CHRNB4CHRNA3CHRNA7
SCHEMBL22069053 0.74 CYP1A2 (0.36) CHRNB2CHRNA4CHRNB4CHRNA3CHRNA7
SCHEMBL31351612 0.74 KMT2A (0.37) CHRNB2CHRNA4CHRNB4CHRNA3CHRNA7
SCHEMBL2403645 0.72 TSHR (0.33) CHRNB2CHRNA4CHRNB4CHRNA3CHRNA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009033689-A1 PIPERIDONE DERIVATIVES AND MEDICAL USES THEREOF HEINRICH-PETTE-INSTITUT (DE) 2009-03-19 WO disclosed
EP-2036556-A1 Piperidone derivatives and medical uses thereof Heinrich-Pette-Institut (DE) 2009-03-18 EP disclosed