SCHEMBL4060730

SCHEMBL4060730

C[Si](C)(C)C#CCCCCCCCCC(=O)O

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN7 P35236 5/20 0.60
HMGCR P04035 5/20 0.60
TDP1 Q9NUW8 3/20 0.50
MAPT P10636 2/20 0.50
RECQL P46063 2/20 0.50
CYP1A2 P05177 1/20 0.50
CYP2D6 P10635 1/20 0.50
CYP2C9 P11712 1/20 0.50
CYP2C19 P33261 1/20 0.50
HSD17B10 Q99714 1/20 0.50
TSHR P16473 2/20 0.48
LMNA P02545 1/20 0.48
NFKB1 P19838 1/20 0.48
PMP22 Q01453 1/20 0.48
EPHX2 P34913 2/20 0.47
ALDH1A1 P00352 2/20 0.47
KDM4E B2RXH2 1/20 0.47
MEN1 O00255 1/20 0.47
USP2 O75604 1/20 0.47
POLB P06746 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9551566 1.00 PTPN7 (0.60) PTPN7HMGCRTDP1MAPTRECQL
SCHEMBL31682050 1.00 PTPN7 (0.60) PTPN7HMGCRTDP1MAPTRECQL
SCHEMBL22029362 1.00 PTPN7 (0.60) PTPN7HMGCRTDP1MAPTRECQL
SCHEMBL4063611 1.00 PTPN7 (0.60) PTPN7HMGCRTDP1MAPTRECQL
SCHEMBL31682065 1.00 PTPN7 (0.60) PTPN7HMGCRTDP1MAPTRECQL
SCHEMBL710828 0.98 PTPN7 (0.57) PTPN7HMGCRTDP1MAPTRECQL
SCHEMBL7315206 0.92 PTPN7 (0.50) PTPN7HMGCRTDP1MAPTRECQL
SCHEMBL6272882 0.83 EPHX2 (0.38) PTPN7HMGCRTDP1MAPTRECQL
SCHEMBL21099048 0.82 HMGCR (0.43) PTPN7HMGCRTDP1MAPTRECQL
SCHEMBL9262800 0.82 PAOX (0.40) PTPN7HMGCRTDP1MAPTRECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2059496-A1 ACETYLENIC COMPOUNDS Commonwealth Scientific and Industrial Research Organisation (AU) 2009-05-20 EP disclosed
WO-2008031157-A1 ACETYLENIC COMPOUNDS COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2008-03-20 WO disclosed
EP-0525479-B1 Spicamycin derivatives and the use thereof KIRIN BREWERY (JP) 1997-11-05 EP disclosed
US-5631238-A ANTICARCINOGENIC AGENTS KIRIN BEER KABUSHIKI KAISHA (JP) 1997-05-20 US disclosed
US-5461036-A Treating colon, gastric, esophageal cancer KIRIN BEER KABUSHIKI KAISHA (JP) 1995-10-24 US disclosed
EP-0525479-A1 Spicamycin derivatives and the use thereof KIRIN BEER KABUSHIKI KAISHA (JP) 1993-02-03 EP disclosed