SCHEMBL4060809

SCHEMBL4060809

CSCCn1c(=O)c2[nH]c(-c3ccc(S(=O)(=O)N4CCN(Cc5ccc(Br)cc5)CC4)cc3)cc2n(CCSC)c1=O

nearest known ligand 0.72

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 19/20 0.72
ADORA1 P30542 13/20 0.72
ADORA3 P0DMS8 10/20 0.72
ADORA2A P29274 4/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4049560 0.91 ADORA2B (0.75) ADORA2BADORA1ADORA3ADORA2A
SCHEMBL4056999 0.89 ADORA2B (0.72) ADORA2BADORA1ADORA3ADORA2A
SCHEMBL4057579 0.88 ADORA2B (0.75) ADORA2BADORA1ADORA3ADORA2A
SCHEMBL4058193 0.85 ADORA2B (0.82) ADORA2BADORA1ADORA3ADORA2A
SCHEMBL4054947 0.85 ADORA2B (0.82) ADORA2BADORA1ADORA3ADORA2A
SCHEMBL4052662 0.84 ADORA2B (1.00) ADORA2BADORA1ADORA3ADORA2A
SCHEMBL4054089 0.83 ADORA2B (0.73) ADORA2BADORA1ADORA3ADORA2A
SCHEMBL4060452 0.83 ADORA2B (0.81) ADORA2BADORA1ADORA3ADORA2A
SCHEMBL4051717 0.83 ADORA2B (0.75) ADORA2BADORA1ADORA3ADORA2A
SCHEMBL4050980 0.82 ADORA2B (0.75) ADORA2BADORA1ADORA3ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7504398-B2 potent and selective antagonists of adenosine receptors; Parkinson's disease, asthma, allergies, inflammation, atherosclerosis, hypertension, gastrointestinal disorders, cell proliferation and autoimmune diseases; sulfonamidation LABORATORIOS ALMIRALL S.A. (ES) 2009-03-17 US disclosed
EP-1492793-B1 NEW-4-(PYRROLOPYRIMIDIN-6-YL)BENZENESULPHONAMIDE DERIVATIVES ALMIRALL LAB (ES) 2008-01-16 EP disclosed