SCHEMBL4060883

SCHEMBL4060883

O=C(O)Cc1c[nH]c2cccc(OCCCOc3ccnc4cc(C(F)(F)F)ccc34)c12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 2/20 0.41
KDM4E B2RXH2 1/20 0.41
MEN1 O00255 1/20 0.41
ALDH1A1 P00352 1/20 0.41
POLB P06746 1/20 0.41
GAA P10253 1/20 0.41
MAPT P10636 1/20 0.41
THRB P10828 1/20 0.41
DNMT1 P26358 1/20 0.41
RECQL P46063 1/20 0.41
CASP6 P55212 1/20 0.41
KMT2A Q03164 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
ITK Q08881 2/20 0.37
SSTR1 P30872 1/20 0.37
SSTR3 P32745 1/20 0.37
HTR1A P08908 1/20 0.37
SLC6A4 P31645 1/20 0.37
TACR1 P25103 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4061859 0.82 MCL1 (0.42) MCL1KDM4EMEN1ALDH1A1POLB
SCHEMBL5012504 0.73 PPARG (0.54) PPARGPPARDPPARAPTGDR2
SCHEMBL28666661 0.72 PTGDR2 (0.53) PRKD3MAP4K4KDRGSK3AGSK3B
SCHEMBL5617095 0.72 KDM4E (0.40) MCL1KDM4EMEN1ALDH1A1POLB
SCHEMBL6052560 0.71 PPARD (0.54) MAPTPPARGPPARDPPARA
SCHEMBL4055211 0.71 NR1H3 (0.65) PPARGPPARDPPARA
SCHEMBL4063165 0.70 GAA (0.48) MCL1KDM4EMEN1ALDH1A1POLB
SCHEMBL6052553 0.70 PPARD (0.54) PPARGPPARDPPARA
SCHEMBL20595203 0.70 CLK4 (0.43) ALDH1A1ITKADRB2PRKD3MAP4K4
Trifluoroacetic Acid SCHEMBL20595199 0.70 GSK3A (0.41) ADRB2PRKD3MAP4K4MARK3KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1689389-A4 INDOLE COMPOUNDS NAT HEALTH RESEARCH INSTITUTES (TW) 2009-06-17 EP disclosed
EP-1689389-A2 INDOLE COMPOUNDS National Health Research Institutes (TW) 2006-08-16 EP disclosed
WO-2005056522-A2 INDOLE COMPOUNDS NATIONAL HEALTH RESEARCH INSTITUTES (TW) 2005-06-23 WO disclosed