SCHEMBL4065156

SCHEMBL4065156

CN(c1ncnc2cc(-c3ccccc3)sc12)C1CCCCC1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 1/20 0.50
FLT1 P17948 3/20 0.47
EGFR P00533 2/20 0.47
CAMKK2 Q96RR4 1/20 0.47
TP53 P04637 2/20 0.46
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
POLB P06746 1/20 0.44
CHEK1 O14757 1/20 0.44
KCNH2 Q12809 1/20 0.44
LMNA P02545 1/20 0.44
JAK1 P23458 3/20 0.43
JAK3 P52333 3/20 0.43
JAK2 O60674 1/20 0.43
GBA1 P04062 3/20 0.42
MAPT P10636 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4073207 0.74 IKBKB (0.53) IKBKBFLT1EGFRTP53POLB
SCHEMBL4070018 0.71 IKBKB (0.50) IKBKBFLT1EGFRKMT2APOLB
SCHEMBL4065154 0.71 FLT1 (0.55) IKBKBFLT1EGFRCAMKK2
SCHEMBL16281232 0.70 IKBKB (0.67) IKBKBFLT1EGFRKMT2ALMNA
SCHEMBL2369031 0.69 LMNA (0.55) FLT1TP53MEN1KMT2APOLB
SCHEMBL3542881 0.69 CSF1R (0.71) EGFRJAK1JAK3JAK2
SCHEMBL4069658 0.69 EGFR (0.47) IKBKBFLT1EGFRMEN1KMT2A
SCHEMBL9056996 0.68 KDM4E (0.40) TP53MEN1KMT2ALMNAJAK3
SCHEMBL4074719 0.68 EGFR (0.46) IKBKBFLT1EGFRPOLBLMNA
SCHEMBL2879120 0.68 NPC1 (0.67) IKBKBFLT1EGFRCAMKK2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090042878-A1 THIENOPYRIMIDYLAMINES AS MODULATORS OF THE EP2 RECEPTOR BAYER SHERING PHARMA AG (DE) 2009-02-12 US claimed
EP-2014663-A1 Thieno-pyrimidyl amines as modulators of EP2 receptors Bayer Schering Pharma AG (DE) 2009-01-14 EP claimed
US-20090042878-A1 THIENOPYRIMIDYLAMINES AS MODULATORS OF THE EP2 RECEPTOR BAYER SHERING PHARMA AG (DE) 2009-02-12 US disclosed
EP-2014663-A1 Thieno-pyrimidyl amines as modulators of EP2 receptors Bayer Schering Pharma AG (DE) 2009-01-14 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090042878-A1 THIENOPYRIMIDYLAMINES AS MODULATORS OF THE EP2 RECEPTOR PTGER2, PTGER1, PTGDR2 IKBKB 2889/4885FLT1 3521/4885EGFR 875/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.