SCHEMBL4066322

SCHEMBL4066322

COc1cccc2c(N3CCN(CCNCc4cc5c(cn4)OCCO5)CC3)c(Cl)cnc12

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SLC2A1 P11166 2/20 0.44
KCNH2 Q12809 8/20 0.43
LMNA P02545 3/20 0.39
MAPT P10636 3/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
KDM4E B2RXH2 2/20 0.39
TDP1 Q9NUW8 1/20 0.39
ALDH1A1 P00352 1/20 0.39
DRD2 P14416 1/20 0.37
DRD4 P21917 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
GLA P06280 1/20 0.37
HTT P42858 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4064313 0.83 KCNH2 (0.53) SLC2A1KCNH2
SCHEMBL4062218 0.83 SLC2A1 (0.47) SLC2A1KCNH2DRD2DRD4
SCHEMBL4062214 0.81 KCNH2 (0.61) KCNH2
SCHEMBL4066049 0.79 KCNH2 (0.43) KCNH2DRD2
SCHEMBL4068256 0.74 KCNH2 (0.35) KCNH2LMNAMAPTKDM4EGLA
SCHEMBL4074226 0.70 SLC2A1 (0.45) SLC2A1KCNH2
SCHEMBL4066607 0.70 KCNH2 (0.54) KCNH2
SCHEMBL4067565 0.70 KCNH2 (0.53) SLC2A1KCNH2
SCHEMBL4074224 0.68 KCNH2 (0.58) KCNH2
SCHEMBL4067925 0.64 KCNH2 (0.49) KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1605938-B1 Antibacterial derivatives of napthydrin and quinoline GLAXO GROUP LTD (GB) 2009-02-11 EP claimed