SCHEMBL4066917

SCHEMBL4066917

CCN(O)S(=O)(=O)c1ccc(Nc2ncc(Br)c(NCCCC(=O)OC)n2)cc1

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CA2 P00918 3/20 0.48
TBK1 Q9UHD2 2/20 0.47
CDK1 P06493 16/20 0.47
CDK2 P24941 15/20 0.47
KDR P35968 15/20 0.47
STK17B O94768 1/20 0.46
STK17A Q9UEE5 1/20 0.46
CCNB1 P14635 2/20 0.44
CCNE1 P24864 2/20 0.44
CDK4 P11802 2/20 0.44
CDK7 P50613 2/20 0.44
CDK9 P50750 2/20 0.44
CCNT1 O60563 1/20 0.44
CCND1 P24385 1/20 0.44
CCNH P51946 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4063585 0.83 CA2 (0.61) CA2TBK1CDK1CDK2KDR
SCHEMBL4066912 0.83 SYK (0.51) CA2TBK1CDK1CDK2KDR
SCHEMBL3865508 0.81 CA2 (0.60) CA2TBK1CDK1CDK2KDR
SCHEMBL4065623 0.80 CA2 (0.57) CA2TBK1CDK1CDK2KDR
SCHEMBL4068494 0.80 CA2 (0.55) CA2TBK1CDK1CDK2KDR
SCHEMBL4061057 0.79 CDK1 (0.55) CA2CDK1CDK2KDRCCNB1
SCHEMBL6448921 0.77 CA2 (0.65) CA2TBK1CDK1CDK2KDR
SCHEMBL4064363 0.76 CDK1 (0.55) CA2CDK1CDK2KDRCCNB1
SCHEMBL3874620 0.76 CA2 (0.64) CA2TBK1CDK1CDK2KDR
SCHEMBL13648585 0.76 CA2 (0.55) CA2TBK1CDK1CDK2KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1392662-B1 CDK INHIBITING PYRIMIDINES, PRODUCTION THEREOF AND THEIR USE AS MEDICAMENTS BAYER SCHERING PHARMA AG (DE) 2009-01-07 EP claimed
EP-1392662-B1 CDK INHIBITING PYRIMIDINES, PRODUCTION THEREOF AND THEIR USE AS MEDICAMENTS BAYER SCHERING PHARMA AG (DE) 2009-01-07 EP disclosed