SCHEMBL4067280

SCHEMBL4067280

CC(C)(C)OC(=O)N1C[C@H]2CC2C1CNCc1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 1/20 0.41
JAK1 P23458 1/20 0.41
ATM Q13315 1/20 0.41
NR1H2 P55055 2/20 0.40
NR1H3 Q13133 2/20 0.40
HDAC8 Q9BY41 1/20 0.39
STS P08842 1/20 0.39
ACHE P22303 1/20 0.39
KDM4E B2RXH2 1/20 0.39
PKM P14618 1/20 0.39
NAMPT P43490 1/20 0.39
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA7 P43166 1/20 0.39
CA14 Q9ULX7 1/20 0.39
ABCB1 P08183 1/20 0.39
KMT2A Q03164 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
KEAP1 Q14145 1/20 0.38
NFE2L2 Q16236 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1338962 1.00 JAK2 (0.41) JAK2JAK1ATMNR1H2NR1H3
SCHEMBL2933059 1.00 JAK2 (0.41) JAK2JAK1ATMNR1H2NR1H3
SCHEMBL2933063 1.00 JAK2 (0.41) JAK2JAK1ATMNR1H2NR1H3
SCHEMBL496466 0.94 JAK2 (0.39) JAK2JAK1ATMNR1H2NR1H3
SCHEMBL496187 0.88 KMT2A (0.41) JAK2JAK1ATMNR1H2NR1H3
SCHEMBL29997881 0.85 NR1H2 (0.48) JAK2JAK1NR1H2NR1H3STS
SCHEMBL29997304 0.85 NR1H2 (0.48) JAK2JAK1NR1H2NR1H3STS
SCHEMBL25678532 0.80 LMNA (0.49) ABCB1L3MBTL1KEAP1NFE2L2LMNA
SCHEMBL3636540 0.78 HTT (0.40) HDAC8KMT2AL3MBTL1DPP4LMNA
SCHEMBL15600175 0.78 NR1H2 (0.37) NR1H2NAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2079690-A2 3-AZA-BICYCLO[3.1.0]HEXANE DERIVATIVES Actelion Pharmaceuticals Ltd. (CH) 2009-07-22 EP disclosed
WO-2008038251-A2 3-AZA-BICYCLO[3.1.0]HEXANE DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2008-04-03 WO disclosed