SCHEMBL4068013

SCHEMBL4068013

[CH](CNCc1ccncc1)Cc1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC2A4 P14672 1/20 0.46
ALDH1A1 P00352 1/20 0.45
GAA P10253 1/20 0.45
MAPT P10636 1/20 0.45
CA9 Q16790 1/20 0.44
HTT P42858 1/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
DPP7 Q9UHL4 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.42
LMNA P02545 1/20 0.42
LSS P48449 1/20 0.42
ROCK2 O75116 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
KCNH3 Q9ULD8 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4065565 0.89 MEN1 (0.54) GAAMAPTMEN1KMT2ATDP1
SCHEMBL4072842 0.83 CYP1A2 (0.62) ALDH1A1HTTCYP1A2CYP2D6
SCHEMBL4068318 0.83 CYP1A2 (0.58) ALDH1A1HTTTDP1CYP1A2CYP2D6
SCHEMBL1042566 0.81 SLC2A4 (0.63) SLC2A4ALDH1A1GAAMAPTCA9
SCHEMBL4067663 0.77 CHRM2 (0.50) ALDH1A1GAAMAPTMEN1KMT2A
4-Formylpyridine SCHEMBL25376714 0.74 SLC2A4 (0.51) SLC2A4ALDH1A1GAAMAPTHTT
SCHEMBL25697049 0.74 ALDH1A1 (0.46) SLC2A4ALDH1A1GAAMAPTHTT
SCHEMBL6616250 0.74 MAOB (0.65) GAAMAPTMEN1KMT2ATDP1
Pyridine SCHEMBL9737571 0.73 CYP1A2 (0.61) SLC2A4ALDH1A1GAAMAPTHTT
SCHEMBL28188921 0.73 GAA (0.74) ALDH1A1GAAMAPTCA9MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1415986-B1 SPIRO ISOBENZOFURANES AS NEUROPEPTIDE Y RECEPTOR ANTAGONISTS BANYU PHARMA CO LTD (JP) 2009-04-08 EP disclosed
US-7205417-B2 Spiro compounds BANYU PHARMACEUTICAL CO., LTD. (JP) 2007-04-17 US disclosed
CN-1538956-A Spiro compounds ������ҩ��ʽ���� 2004-10-20 CN disclosed