SCHEMBL4068658

SCHEMBL4068658

CCc1ccc(F)cc1C(=O)N[C@@H](Cc1ccc(OCCc2ccc3c(n2)OCCN3)cc1)C(=O)O

nearest known ligand 0.57

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 18/20 0.57
ITGA5 P08648 18/20 0.57
ITGB3 P05106 17/20 0.57
ITGAV P06756 16/20 0.57
ITGA2B P08514 1/20 0.40
PPARG P37231 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4068793 0.94 ITGB1 (0.65) ITGB1ITGA5ITGB3ITGAVITGA2B
SCHEMBL4068084 0.91 ITGB1 (0.58) ITGB1ITGA5ITGB3ITGAV
SCHEMBL4929434 0.89 ITGB1 (0.68) ITGB1ITGA5ITGB3ITGAVITGA2B
SCHEMBL4069743 0.83 ITGB1 (0.58) ITGB1ITGA5ITGB3ITGAV
SCHEMBL4743659 0.83 ITGB1 (0.54) ITGB1ITGA5ITGB3ITGAVPPARG
SCHEMBL4068227 0.83 ITGB1 (0.63) ITGB1ITGA5ITGB3ITGAVITGA2B
SCHEMBL4066312 0.83 ITGB1 (0.65) ITGB1ITGA5ITGB3ITGAV
SCHEMBL4924731 0.83 ITGB3 (0.68) ITGB1ITGA5ITGB3ITGAVITGA2B
SCHEMBL4074983 0.82 ITGB1 (0.64) ITGB1ITGA5ITGB3ITGAV
SCHEMBL4073721 0.81 ITGB1 (0.59) ITGB1ITGA5ITGB3ITGAV

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2049490-A1 N-(BENZOYL)-O- [2- (PYRIDIN- 2 -YLAMINO) ETHYL]-L-TYROSINE DERIVATIVES AND RELATED COMPOUNDS AS A5B1 ANTAGONISTS FOR THE TREATMENT OF SOLID TUMORS Astra Zeneca AB (SE) 2009-04-22 EP claimed
WO-2007141473-A1 N-(BENZOYL)-O- [2- (PYRIDIN- 2 -YLAMINO) ETHYL] -L-TYROSINE DERIVATIVES AND RELATED COMPOUNDS AS A5B1 ANTAGONISTS FOR THE TREATMENT OF SOLID TUMORS ASTRAZENECA AB (SE) 2007-12-13 WO claimed
EP-2049490-A1 N-(BENZOYL)-O- [2- (PYRIDIN- 2 -YLAMINO) ETHYL]-L-TYROSINE DERIVATIVES AND RELATED COMPOUNDS AS A5B1 ANTAGONISTS FOR THE TREATMENT OF SOLID TUMORS Astra Zeneca AB (SE) 2009-04-22 EP disclosed
WO-2007141473-A1 N-(BENZOYL)-O- [2- (PYRIDIN- 2 -YLAMINO) ETHYL] -L-TYROSINE DERIVATIVES AND RELATED COMPOUNDS AS A5B1 ANTAGONISTS FOR THE TREATMENT OF SOLID TUMORS ASTRAZENECA AB (SE) 2007-12-13 WO disclosed