SCHEMBL4070229

SCHEMBL4070229

NS(=O)(=O)c1ccc(Nc2ncc(Br)c(NC3CCOC3)n2)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SYK P43405 6/20 0.58
IGF1R P08069 2/20 0.55
CA2 P00918 4/20 0.54
CDK1 P06493 6/20 0.53
KDR P35968 6/20 0.53
CDK2 P24941 5/20 0.53
CDK4 P11802 2/20 0.53
CDK7 P50613 2/20 0.53
CDK9 P50750 2/20 0.53
CCNT1 O60563 1/20 0.53
CCND1 P24385 1/20 0.53
CCNH P51946 1/20 0.53
CCNB1 P14635 1/20 0.52
CCNE1 P24864 1/20 0.52
PTK2 Q05397 2/20 0.48
NUAK1 O60285 1/20 0.46
STK16 O75716 1/20 0.46
NTRK1 P04629 1/20 0.46
CSF1R P07333 1/20 0.46
CSNK2A2 P19784 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4070220 1.00 SYK (0.58) SYKIGF1RCA2CDK1KDR
SCHEMBL4058413 0.85 SYK (0.69) SYKIGF1RCA2CDK1KDR
SCHEMBL4064533 0.85 SYK (0.69) SYKIGF1RCA2CDK1KDR
SCHEMBL4068789 0.85 SYK (0.68) SYKIGF1RCA2CDK1KDR
SCHEMBL4580306 0.84 CDK1 (0.44) SYKIGF1RCA2CDK1KDR
SCHEMBL14000045 0.84 CDK1 (0.44) SYKIGF1RCA2CDK1KDR
SCHEMBL4070462 0.83 SYK (0.69) SYKIGF1RCA2CDK1KDR
SCHEMBL4068613 0.83 SYK (0.62) SYKIGF1RCA2CDK1KDR
SCHEMBL14498929 0.83 SYK (0.69) SYKIGF1RCA2CDK1KDR
SCHEMBL13648587 0.83 SYK (0.69) SYKIGF1RCA2CDK1KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1392662-B1 CDK INHIBITING PYRIMIDINES, PRODUCTION THEREOF AND THEIR USE AS MEDICAMENTS BAYER SCHERING PHARMA AG (DE) 2009-01-07 EP claimed
EP-1392662-B1 CDK INHIBITING PYRIMIDINES, PRODUCTION THEREOF AND THEIR USE AS MEDICAMENTS BAYER SCHERING PHARMA AG (DE) 2009-01-07 EP disclosed