SCHEMBL4071291

SCHEMBL4071291

CC(C)(C(=O)Nc1cc2ccccc2cn1)S(=O)(=O)c1ccc(Cl)cc1.CC(C)(C(=O)Nc1nc(-c2ccccc2)ns1)S(=O)(=O)c1ccc(Cl)cc1.Cn1nc(C2CC2)cc1NC(=O)C(C)(C)S(=O)(=O)c1ccc(Cl)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 9/20 0.46
CNR1 P21554 6/20 0.43
TP53 P04637 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
NPC1 O15118 1/20 0.40
LMNA P02545 1/20 0.40
POLB P06746 1/20 0.40
NFKB1 P19838 1/20 0.40
RAB9A P51151 1/20 0.40
NFKB2 Q00653 1/20 0.40
RELA Q04206 1/20 0.40
ADORA3 P0DMS8 4/20 0.38
USP36 Q9P275 1/20 0.38
ALOX15 P16050 1/20 0.36
MAPK1 P28482 1/20 0.36
CASP1 P29466 1/20 0.36
CASP7 P55210 1/20 0.36
HSD17B10 Q99714 1/20 0.36
WNT1 P04628 1/20 0.35
GSK3B P49841 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4069777 0.94 CNR2 (0.42) CNR2CNR1TP53SMN1; SMN2NPC1
SCHEMBL1464390 0.79 CNR2 (0.71) CNR2CNR1CYP3A4GAACYP2C19
SCHEMBL1465115 0.78 SMN1; SMN2 (0.65) CNR2CNR1TP53SMN1; SMN2NPC1
SCHEMBL3961157 0.77 CNR2 (0.40) CNR2CNR1NPC1RAB9AMAPK1
SCHEMBL1463634 0.76 CNR2 (0.66) CNR2CNR1
SCHEMBL3962989 0.76 CNR2 (0.53) CNR2CNR1LMNA
SCHEMBL1465923 0.76 CNR2 (0.68) CNR2CNR1LMNACYP3A4GAA
SCHEMBL3964882 0.75 CNR2 (0.67) CNR2CNR1LMNACYP3A4GAA
SCHEMBL1465913 0.75 CNR2 (0.67) CNR2CNR1LMNACYP3A4GAA
SCHEMBL4064491 0.74 MEN1 (0.52) CNR2CNR1TP53SMN1; SMN2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2081905-A2 SULFONYL COMPOUNDS WHICH MODULATE THE CB2 RECEPTOR Boehringer Ingelheim International GmbH (DE) 2009-07-29 EP disclosed
WO-2008014199-A2 SULFONYL COMPOUNDS WHICH MODULATE THE CB2 RECEPTOR BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-01-31 WO disclosed