SCHEMBL4073145

SCHEMBL4073145

Cc1nc(Cl)nc(Nc2cc(C3CC3)[nH]n2)c1Br

nearest known ligand 0.54

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
IGF1R P08069 20/20 0.54
NTRK1 P04629 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL56235 0.80 IGF1R (0.54) IGF1RNTRK1
SCHEMBL2317829 0.80 IGF1R (0.75) IGF1RNTRK1
SCHEMBL1164462 0.80 IGF1R (0.66) IGF1RNTRK1
SCHEMBL2321718 0.77 IGF1R (0.68) IGF1R
SCHEMBL4071502 0.77 NTRK1 (0.61) IGF1RNTRK1
SCHEMBL14606170 0.77 IGF1R (0.45) IGF1RNTRK1
SCHEMBL4068008 0.77 NTRK1 (0.61) NTRK1
SCHEMBL2319952 0.77 PIK3C3 (0.55) IGF1R
SCHEMBL3006826 0.76 IGF1R (0.56) IGF1R
SCHEMBL219252 0.76 IGF1R (0.66) IGF1RNTRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1686999-B1 PYRAZOLE DERIVATIVES AS INHIBITORS OF RECEPTOR TYROSINE KINASES ASTRAZENECA AB (SE) 2009-07-01 EP disclosed