SCHEMBL4073323

SCHEMBL4073323

CC1(N2CCC(c3ccccc3)CC2)CCN(C(N)C=O)C1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CSNK1D P48730 1/20 0.39
CSNK1G2 P78368 1/20 0.39
KCNH2 Q12809 2/20 0.38
HRH3 Q9Y5N1 1/20 0.38
SLC18A3 Q16572 3/20 0.38
CCR5 P51681 5/20 0.36
DRD2 P14416 1/20 0.35
NR1H2 P55055 1/20 0.35
NR1H3 Q13133 1/20 0.35
HSD11B1 P28845 2/20 0.34
HTR7 P34969 2/20 0.34
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA7 P43166 1/20 0.34
CA9 Q16790 1/20 0.34
CA14 Q9ULX7 1/20 0.34
CARM1 Q86X55 1/20 0.33
PRMT6 Q96LA8 1/20 0.33
OPRM1 P35372 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8891712 0.79 KCNH2 (0.46) KCNH2HRH3SLC18A3DRD2CA12
SCHEMBL27764392 0.74 CSNK1D (0.52) CSNK1DCSNK1G2KCNH2HRH3SLC18A3
SCHEMBL4881149 0.71 CSNK1D (0.55) CSNK1DCSNK1G2KCNH2HRH3SLC18A3
SCHEMBL4070366 0.70 SLC18A3 (0.49) SLC18A3
SCHEMBL27498942 0.68 KCNH2 (0.52) KCNH2HRH3SLC18A3CCR5DRD2
SCHEMBL4071190 0.68 NAMPT (0.48) CSNK1DCSNK1G2CCR5
SCHEMBL4076805 0.66 SLC18A3 (0.46) SLC18A3CCR5DRD2CARM1PRMT6
SCHEMBL24291907 0.65 KCNH2 (0.53) KCNH2HRH3SLC18A3CCR5DRD2
SCHEMBL3710421 0.63 SLC18A3 (0.52) SLC18A3DRD2CARM1PRMT6
SCHEMBL16255639 0.63 KCNH2 (0.54) KCNH2HRH3SLC18A3DRD2CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2099454-A2 AMINOPYRROLIDINES AS CHEMOKINE RECEPTOR ANTAGONISTS Abbott Laboratories (US) 2009-09-16 EP disclosed
WO-2008060621-A2 AMINOPYRROLIDINES AS CHEMOKINE RECEPTOR ANTAGONISTS ABBOTT LABORATORIES (US) 2008-05-22 WO disclosed