SCHEMBL4078672

SCHEMBL4078672

CC(C)Oc1ccc2c(Cl)nc(OC(=O)O)c(O)c2c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.39
KMT2A Q03164 4/20 0.38
KDM4E B2RXH2 3/20 0.37
HPGD P15428 3/20 0.37
LMNA P02545 3/20 0.37
GAA P10253 2/20 0.37
MCL1 Q07820 1/20 0.37
EGLN1 Q9GZT9 5/20 0.36
THRA P10827 1/20 0.36
THRB P10828 1/20 0.36
PRKAB2 O43741 1/20 0.36
PRKAG1 P54619 1/20 0.36
PRKAA2 P54646 1/20 0.36
PRKAA1 Q13131 1/20 0.36
PRKAG3 Q9UGI9 1/20 0.36
PRKAG2 Q9UGJ0 1/20 0.36
PRKAB1 Q9Y478 1/20 0.36
BBOX1 O75936 2/20 0.36
FTO Q9C0B1 1/20 0.36
MEN1 O00255 3/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4078616 0.95 EGLN1 (0.41) ALDH1A1KMT2AKDM4EHPGDLMNA
SCHEMBL4075081 0.87 DHODH (0.44) ALDH1A1KDM4EHPGDLMNAEGLN1
SCHEMBL1033757 0.82 SCN9A (0.35) ALDH1A1KDM4EHPGDLMNAGAA
SCHEMBL4078497 0.82 ESR1 (0.38) ALDH1A1KMT2AKDM4EHPGDLMNA
SCHEMBL1033120 0.82 SMN1; SMN2 (0.47) ALDH1A1EGLN1THRATHRBPRKAB2
SCHEMBL522422 0.82 EGLN1 (0.45) ALDH1A1KMT2AKDM4EHPGDLMNA
SCHEMBL4069669 0.82 DHODH (0.44) ALDH1A1KDM4EHPGDLMNAEGLN1
SCHEMBL4074682 0.81 DHODH (0.39) ALDH1A1KMT2AGAAMEN1TP53
SCHEMBL1034732 0.81 NPC1 (0.38) EGLN1THRATHRBNPC1RAB9A
SCHEMBL1031021 0.80 NPC1 (0.38) ALDH1A1KDM4EHPGDLMNAEGLN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1538160-B1 Substituted Isoquinolin-3-carboxyamides, their preparation and medical use FIBROGEN INC (US) 2009-06-03 EP disclosed