SCHEMBL4083284

SCHEMBL4083284

Cc1cn(C)c2ccc(-n3c(S)nnc3-c3cc(C(C)C)cc(O)c3O)cc12

nearest known ligand 0.36

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 17/20 0.36
HSP90AB1 P08238 17/20 0.36
TRPA1 O75762 1/20 0.32
PTGS1 P23219 1/20 0.32
CACNA1C Q13936 1/20 0.32
HSP90B1 P14625 1/20 0.30
TRAP1 Q12931 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL421461 0.84 HSP90AA1 (0.52) HSP90AA1HSP90AB1HSP90B1TRAP1
SCHEMBL421199 0.78 HSP90AA1 (0.35) HSP90AA1HSP90AB1
SCHEMBL419020 0.78 HSP90AA1 (0.38) HSP90AA1HSP90AB1HSP90B1TRAP1
SCHEMBL4088362 0.75 MAP3K11 (0.37) HSP90AA1HSP90AB1
SCHEMBL419166 0.73 HSP90AA1 (0.53) HSP90AA1HSP90AB1HSP90B1TRAP1
SCHEMBL421098 0.73 HSP90AA1 (0.45) HSP90AA1HSP90AB1HSP90B1TRAP1
SCHEMBL3989106 0.72 HSP90AA1 (0.55) HSP90AA1HSP90AB1HSP90B1TRAP1
SCHEMBL419851 0.70 HSP90AA1 (0.40) HSP90AA1HSP90AB1HSP90B1TRAP1
SCHEMBL3301787 0.69 HSP90AA1 (0.40) HSP90AA1HSP90AB1HSP90B1TRAP1
SCHEMBL3301790 0.69 HSP90AA1 (0.40) HSP90AA1HSP90AB1HSP90B1TRAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2054059-A2 TRIAZOLE COMPOUNDS THAT MODULATE HSP90 ACTIVITY Synta Pharmaceuticals Corporation (US) 2009-05-06 EP disclosed
WO-2008021364-A2 TRIAZOLE COMPOUNDS THAT MODULATE HSP90 ACTIVITY SYNTA PHARMACEUTICALS CORP. (US) 2008-02-21 WO disclosed