SCHEMBL4086058

SCHEMBL4086058

COc1cc(C(=O)c2cn(C(C)C)c3ncnc(N)c23)cc(NS(=O)(=O)c2ccccc2F)n1

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 4/20 0.50
NTRK2 Q16620 3/20 0.50
NTRK3 Q16288 2/20 0.50
KCNH2 Q12809 3/20 0.49
EIF2AK3 Q9NZJ5 1/20 0.47
PDPK1 O15530 8/20 0.47
PDGFRB P09619 1/20 0.46
RET P07949 4/20 0.42
EGFR P00533 2/20 0.42
ERBB2 P04626 2/20 0.42
ERBB3 P21860 2/20 0.42
TEK Q02763 2/20 0.42
ERBB4 Q15303 2/20 0.42
LCK P06239 2/20 0.41
SRC P12931 2/20 0.41
AKT1 P31749 5/20 0.41
MTOR P42345 5/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4086042 0.90 NTRK1 (0.52) NTRK1NTRK2NTRK3KCNH2EIF2AK3
SCHEMBL4076485 0.86 NTRK1 (0.64) NTRK1NTRK2NTRK3KCNH2EIF2AK3
SCHEMBL4085582 0.85 NTRK1 (0.65) NTRK1NTRK2NTRK3KCNH2EIF2AK3
SCHEMBL1942841 0.84 EIF2AK3 (0.53) NTRK1NTRK2NTRK3KCNH2EIF2AK3
SCHEMBL4081490 0.82 PDPK1 (0.55) NTRK1NTRK2NTRK3KCNH2EIF2AK3
SCHEMBL1939947 0.82 PDGFRB (0.62) NTRK1NTRK2NTRK3KCNH2EIF2AK3
SCHEMBL4080442 0.81 NTRK1 (0.58) NTRK1NTRK2NTRK3KCNH2PDPK1
SCHEMBL4080682 0.79 PDPK1 (0.55) NTRK1NTRK2NTRK3KCNH2PDPK1
SCHEMBL4079511 0.79 NTRK1 (0.49) NTRK1NTRK2NTRK3KCNH2EIF2AK3
SCHEMBL1941376 0.78 EIF2AK3 (0.51) NTRK1NTRK2NTRK3KCNH2EIF2AK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7595325-B2 Substituted pyrrolo[2,3-d]pyrimidine derivatives useful in cancer treatment PFIZER INC. (US) 2009-09-29 US disclosed