Moexipril

Moexipril

SCHEMBL40877

CCOC(=O)[C@H](CCc1ccccc1)N[C@@H](C)C(=O)N1Cc2cc(OC)c(OC)cc2C[C@H]1C(=O)O.Cl

nearest known ligand 0.98

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACE

The experimentally established mechanism targets of Moexipril. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ACE known ✓ P12821 15/20 0.98
PDE3A Q14432 1/20 0.98
ABCB11 O95342 2/20 0.79
LMNA P02545 1/20 0.63
SMN1; SMN2 Q16637 1/20 0.58
AGTR2 P50052 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Moexipril SCHEMBL3967866 1.00 ACE (0.98) ACEPDE3AABCB11LMNASMN1; SMN2
Moexipril SCHEMBL28096307 1.00 ACE (0.98) ACEPDE3AABCB11LMNASMN1; SMN2
Moexipril SCHEMBL30903896 1.00 ACE (0.98) ACEPDE3AABCB11LMNASMN1; SMN2
Moexipril SCHEMBL9809013 1.00 ACE (0.98) ACEPDE3AABCB11LMNASMN1; SMN2
Moexipril SCHEMBL29383460 1.00 ACE (0.98) ACEPDE3AABCB11LMNASMN1; SMN2
Moexipril SCHEMBL14660386 1.00 ACE (0.98) ACEPDE3AABCB11LMNASMN1; SMN2
Moexipril SCHEMBL5386742 1.00 ACE (0.98) ACEPDE3AABCB11LMNASMN1; SMN2
Moexipril SCHEMBL11268790 0.99 ACE (0.97) ACEPDE3AABCB11LMNASMN1; SMN2
Moexipril SCHEMBL683321 0.99 ACE (1.00) ACEPDE3AABCB11LMNASMN1; SMN2
Moexipril SCHEMBL22175779 0.99 ACE (1.00) ACEPDE3AABCB11LMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 3984 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4691556-A2 HUMANIZED ANTI-ACTH ANTIBODIES AND USE THEREOF H. Lundbeck A/S (DK) 2026-02-11 EP claimed
US-20230174641-A1 ANTI-ACTH ANTIBODIES AND USE THEREOF H LUNDBECK AS (DK) 2023-06-08 US claimed
US-20230134521-A1 COMPOUNDS FOR METHODS FOR PROMOTING FEMALE REPRODUCTIVE HEALTH THROUGH MEDIATION OF RENIN ANGIOTENSIN FUNCTION SHANAHAN MICHAEL EMIL (US) 2023-05-04 US claimed
US-20210198741-A1 IDENTIFICATION OF SPATIAL BIOMARKERS OF HEART DISORDERS AND METHODS OF USING THE SAME 10X GENOMICS, INC. 2021-07-01 US claimed
EP-3835319-A1 HUMANIZED ANTI-ACTH ANTIBODIES AND USE THEREOF Alder Biopharmaceuticals, Inc. (US) 2021-06-16 EP claimed
EP-3753950-A2 ANTI-PCSK9 ANTIBODIES AND USE THEREOF H. Lundbeck A/S (DK) 2020-12-23 EP claimed
US-20200317772-A1 ANTI-ACTH ANTIBODIES AND USE THEREOF ALDERBIO HOLDINGS LLC (US) 2020-10-08 US claimed
US-20190085073-A1 HUMANIZED ANTI-ACTH ANTIBODIES AND USE THEREOF H. LUNDBECK A/S (DK) 2019-03-21 US claimed
US-10154856-B2 Therapeutic substance transfer catheter and method SILLENDER MARK (AU) 2018-12-18 US claimed
US-10149909-B2 Fortifier TORAY INDUSTRIES, INC. (JP) 2018-12-11 US claimed
JP-2003508349-A 2003-03-04 JP claimed
WO-2002058731-A2 COMBINATIONS OF STEROL ABSORPTION INHIBITOR(S) WITH CARDIOVASCULAR AGENT(S) FOR THE TREATMENT OF VASCULAR CONDITIONS SCHERING CORPORATION (US) 2002-08-01 WO claimed
US-20020049155-A1 Cobalamin compounds useful as cardiovascular agents and as imaging agents HOGENKAMP HENRICUS P C (US) 2002-04-25 US claimed
US-20020037858-A1 Pharmaceutical compositions comprising moexipril magnesium APOTEX, INC. (CA) 2002-03-28 US claimed
EP-1183011-A1 METHOD OF TREATING ANGINA AND/OR ANGINAL EQUIVALENTS, AND PHARMACEUTICAL COMPOSITIONS AND KIT RELATED THERETO Esperion Mergerco, Inc. (US) 2002-03-06 EP claimed
WO-2001092283-A2 COBALAMIN COMPOUNDS USEFUL AS CARDIOVASCULAR AGENTS AND AS IMAGING AGENTS MAYO FOUNDATION FOR MEDICAL EDUCATION AND RESEARCH (US) 2001-12-06 WO claimed
EP-1142878-A2 Pharmaceutical compositions comprising moexipril magnesium SHERMAN, Bernard Charles (CA) 2001-10-10 EP claimed
WO-2000069412-A1 METHOD OF TREATING ANGINA AND/OR ANGINAL EQUIVALENTS, AND PHARMACEUTICAL COMPOSITIONS AND KIT RELATED THERETO ESPERION LUV DEVELOPMENT, INC. (US) 2000-11-23 WO claimed
EP-0220107-A2 Use of angiotensin-converting enzyme inhibitors in macular degeneration MERCK & CO. INC. (US) 1987-04-29 EP claimed
US-4656188-A Ace inhibitors in macular degeneration MERCK & CO., INC. (US) 1987-04-07 US claimed