SCHEMBL4089

SCHEMBL4089

CCOC(=O)CC1(c2ccc(-c3ccc(-c4onc(C)c4N(CC)c4cc(-c5ccccc5)no4)cc3)cc2)CC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 2/20 0.39
GAA P10253 1/20 0.38
PTPN1 P18031 2/20 0.35
ALDH1A1 P00352 4/20 0.35
ABCC3 O15438 1/20 0.34
ABCC4 O15439 1/20 0.34
ABCB11 O95342 1/20 0.34
CYP2C8 P10632 1/20 0.34
CYP2C9 P11712 1/20 0.34
ABCB4 P21439 1/20 0.34
LPAR1 Q92633 1/20 0.34
ABCC2 Q92887 1/20 0.34
SLCO1B3 Q9NPD5 1/20 0.34
SLCO1B1 Q9Y6L6 1/20 0.34
IP6K1 Q92551 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
SMN1; SMN2 Q16637 3/20 0.32
MAPT P10636 2/20 0.32
AKT1 P31749 2/20 0.32
AKT2 P31751 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4790 0.92 BRD4 (0.34) BRD4ALDH1A1ABCC3ABCC4ABCB11
SCHEMBL6641 0.84 GAA (0.37) BRD4GAAALDH1A1ABCC3ABCC4
SCHEMBL13437 0.79 LPAR1 (0.44) BRD4GAAPTPN1ALDH1A1ABCC3
SCHEMBL4090 0.77 LPAR1 (0.40) BRD4GAAPTPN1ALDH1A1ABCC3
SCHEMBL7222 0.76 ABCC3 (0.34) BRD4ALDH1A1ABCC3ABCC4ABCB11
SCHEMBL4392 0.75 LPAR1 (0.42) BRD4GAAALDH1A1ABCC3ABCC4
SCHEMBL4183 0.74 GAA (0.42) BRD4GAAALDH1A1ABCC3ABCC4
SCHEMBL6591 0.74 GAA (0.42) BRD4GAAALDH1A1ABCC3ABCC4
SCHEMBL4182 0.74 BRD4 (0.38) BRD4GAAABCC3ABCC4ABCB11
SCHEMBL6411 0.73 BRD4 (0.33) BRD4ALDH1A1ABCC3ABCC4ABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2483251-A2 POLYCYCLIC COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS Amira Pharmaceuticals, Inc. (US) 2012-08-08 EP disclosed
WO-2011041462-A2 POLYCYCLIC COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS AMIRA PHARMACEUTICALS, INC. (US) 2011-04-07 WO disclosed