Morphine

Morphine

SCHEMBL40902

CN1CC[C@]23c4c5ccc(O)c4O[C@H]2[C@@H](O)C=C[C@H]3[C@H]1C5.Cl

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

OPRM1

The experimentally established mechanism targets of Morphine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
OPRM1 known ✓ P35372 8/20 0.98
OPRD1 P41143 11/20 0.98
OPRK1 P41145 7/20 0.98
MRGPRX2 Q96LB1 4/20 0.98
SLC22A1 O15245 1/20 0.98
ADRA2A P08913 1/20 0.98
ARRB1 P49407 1/20 0.98
ADRB1 P08588 1/20 0.74
PDE4D Q08499 1/20 0.74
PDE3A Q14432 1/20 0.74

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Morphine SCHEMBL27598945 1.00 OPRD1 (0.98) OPRD1OPRM1OPRK1MRGPRX2SLC22A1
Morphine SCHEMBL29461927 1.00 OPRD1 (0.98) OPRD1OPRM1OPRK1MRGPRX2SLC22A1
Morphine SCHEMBL8378216 1.00 OPRD1 (0.98) OPRD1OPRM1OPRK1MRGPRX2SLC22A1
Morphine SCHEMBL27706849 0.99 OPRD1 (0.96) OPRD1OPRM1OPRK1MRGPRX2SLC22A1
Morphine SCHEMBL29846325 0.99 OPRD1 (0.96) OPRD1OPRM1OPRK1MRGPRX2SLC22A1
Morphine SCHEMBL14109970 0.99 OPRD1 (0.96) OPRD1OPRM1OPRK1MRGPRX2SLC22A1
Morphine SCHEMBL147362 0.99 OPRD1 (0.96) OPRD1OPRM1OPRK1MRGPRX2SLC22A1
Morphine SCHEMBL24599520 0.99 OPRD1 (1.00) OPRD1OPRM1OPRK1MRGPRX2SLC22A1
Morphine SCHEMBL13154676 0.99 OPRD1 (1.00) OPRD1OPRM1OPRK1MRGPRX2SLC22A1
Morphine SCHEMBL13696339 0.99 OPRD1 (1.00) OPRD1OPRM1OPRK1MRGPRX2SLC22A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 5577 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4602049-A1 SOS1 INHIBITORS Bayer Aktiengesellschaft (DE) 2025-08-20 EP claimed
EP-4587439-A1 SULFONE-SUBSTITUTED PYRIDO[3,4-D]PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF CANCER Bayer Aktiengesellschaft (DE) 2025-07-23 EP claimed
US-20250154170-A1 FUSED PYRIMIDINES AS KRAS INHIBITORS BAYER AKTIENGESELLSCHAFT (DE) 2025-05-15 US claimed
US-12285488-B2 Oral dosage form containing theobromine-free cocoa LTS LOHMANN THERAPIE-SYSTEME AG (DE) 2025-04-29 US claimed
CN-119894893-A Sulfone substituted pyrido [3,4-D ] pyrimidine derivatives for the treatment of cancer 拜耳公司 2025-04-25 CN claimed
WO-2025021997-A1 NEW MAP4K1 INHIBITORS Deutsches Krebsforschungszentrum Stiftung des öffentlichen Rechts (DE) 2025-01-30 WO claimed
WO-2025016899-A1 SPIROCYCLIC COMPOUNDS FOR THE TREATMENT OF CANCER BAYER AKTIENGESELLSCHAFT (DE) 2025-01-23 WO claimed
EP-4476221-A1 FUSED PYRIMIDINES AS KRAS INHIBITORS Bayer Aktiengesellschaft (DE) 2024-12-18 EP claimed
CN-117461602-B Construction method of morphine addiction animal model 六合熙诚(北京)信息科技有限公司 2024-10-25 CN claimed
EP-3706762-B1 N4-HYDROXYCYTIDINE DERIVATIVE AND ANTI-VIRAL USES RELATED THERETO UNIV EMORY (US) 2024-10-16 EP claimed
WO-1994003161-A1 CONTROLLED RELEASE MORPHINE PREPARATION GACELL LABORATORIES AB (SE) 1994-02-17 WO claimed
US-5240932-A In mixture with terpene and an oil Morimoto, Yasunori (JP) 1993-08-31 US claimed
US-5202128-A Oral administering F. H. FAULDING & CO. LIMITED (AU) 1993-04-13 US claimed
US-5102887-A Method for reducing emesis and nausea induced by the administration of an emesis causing agent ARCH DEVELOPMENT CORPORATION (US) 1992-04-07 US claimed
EP-0476205-A1 Sustained release morphine preparation for rectal administration TORII & CO., LTD. (JP) 1992-03-25 EP claimed
US-5061492-A biodegeadeable polymer matrix is copolymer of gylcolic acid a nd lactic acid TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1991-10-29 US claimed
EP-0430414-A1 Morphine hydrochloride preparation for rectal administration TORII & CO., LTD. (JP) 1991-06-05 EP claimed
US-4711782-A Prolonged release microcapsules and their production TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1987-12-08 US claimed
EP-0046270-B1 NOVEL DERIVATIVES OF BIO-AFFECTING PHENOLIC COMPOUNDS AND PHARMACEUTICAL COMPOSITION CONTAINING THEM INTERx RESEARCH CORPORATION (US) 1986-05-21 EP claimed
US-4389404-A POLYVINYLPYRROLIDONE, MORPHINE HYDROCHLORIDE ZHOROV VLADIMOR I (SU) 1983-06-21 US claimed