SCHEMBL409924

SCHEMBL409924

OC(CCl)CCc1ccc(Cl)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 2/20 0.45
IGF1R P08069 1/20 0.44
ALOX15 P16050 1/20 0.44
HTR3E A5X5Y0 1/20 0.41
HTR3B O95264 1/20 0.41
HTR3A P46098 1/20 0.41
HTR3D Q70Z44 1/20 0.41
HTR3C Q8WXA8 1/20 0.41
CYP2D6 P10635 2/20 0.41
HDAC3 O15379 1/20 0.41
HDAC4 P56524 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC7 Q8WUI4 1/20 0.41
HDAC2 Q92769 1/20 0.41
HDAC10 Q969S8 1/20 0.41
HDAC11 Q96DB2 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
HDAC9 Q9UKV0 1/20 0.41
HDAC5 Q9UQL6 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16314688 0.83 TAAR1 (0.45) TAAR1IGF1RALOX15HTR3EHTR3B
SCHEMBL11462575 0.83 TAAR1 (0.45) TAAR1IGF1RALOX15HTR3EHTR3B
SCHEMBL408931 0.82 TAAR1 (0.43) TAAR1MMP2MMP9MMP12MMP13
SCHEMBL10247192 0.82 CYP1A2 (0.43) TAAR1IGF1RALOX15CYP1A2MMP2
SCHEMBL11180436 0.82 TAAR1 (0.43) TAAR1IGF1RALOX15HTR3EHTR3B
SCHEMBL14135335 0.82 TAAR1 (0.44) TAAR1HTR3EHTR3BHTR3AHTR3D
SCHEMBL8371056 0.81 MMP12 (0.49) CYP2D6MMP2MMP9MMP12MMP13
SCHEMBL3769347 0.81 MMP12 (0.49) CYP2D6MMP2MMP9MMP12MMP13
SCHEMBL11062642 0.80 TAAR1 (0.50) TAAR1IGF1RALOX15HTR3EHTR3B
SCHEMBL12517335 0.80 MMP12 (0.53) MMP2MMP9MMP12MMP13MMP14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 44 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105175341-A Method for industrially synthesizing butoconazole nitrate intermediate ZHUZHOU QIANJIN PHARMACEUTICAL CO LTD 2015-12-23 CN claimed
JP-4795973-B2 2011-10-19 JP claimed
CN-101328110-A Preparation of butoconazole nitrate intermediate BEIJING D VENTURE PHARM TECH (CN) 2008-12-24 CN claimed
JP-2007519699-A 2007-07-19 JP claimed
EP-1709005-A1 HIGH PURITY BUTOCONAZOLE NITRATE WITH SPECIFIED PARTICLE SIZE AND A PROCESS FOR PREPARATION THEREOF RICHTER GEDEON VEGYESZETI GYAR RT. (HU) 2006-10-11 EP claimed
WO-2005070897-A1 HIGH PURITY BUTOCONAZOLE NITRATE WITH SPECIFIED PARTICLE SIZE AND A PROCESS FOR PREPARATION THEREOF Richter Gedeon Vegyészeti Gyár Rt. (HU) 2005-08-04 WO claimed
CN-105218455-B A kind of method for industrializing continuous production Butoconazole Nitrate 株洲千金药业股份有限公司 2018-07-03 CN disclosed
CN-105384600-A Industrial production method for butoconazole nitrate intermediate ZHUZHOU QIANJIN PHARMACEUTICAL CO LTD 2016-03-09 CN disclosed
CN-105198708-A Method for industrially producing butoconazole nitrate intermediate ZHUZHOU QIANJIN PHARMACEUTICAL CO LTD 2015-12-30 CN disclosed
CN-105198817-A Method for industrially synthesizing butoconazole nitrate intermediate ZHUZHOU QIANJIN PHARMACEUTICAL CO LTD 2015-12-30 CN disclosed
CN-105175341-A Method for industrially synthesizing butoconazole nitrate intermediate ZHUZHOU QIANJIN PHARMACEUTICAL CO LTD 2015-12-23 CN disclosed
CN-105175341-A Method for industrially synthesizing butoconazole nitrate intermediate ZHUZHOU QIANJIN PHARMACEUTICAL CO LTD 2015-12-23 CN disclosed
CN-103880596-A Preparation method of butoconazole nitrate intermediate suitable for industrial production LING PEIXUE 2014-06-25 CN disclosed
EP-0005980-B1 DERIVATIVES OF SUBSTITUTED N-ALKYL IMIDAZOLES, THEIR PREPARATION AND THESE COMPOUNDS FOR PHARMACEUTICAL USE SYNTEX (U.S.A.) INC. (US) 1984-08-29 EP disclosed
US-4421758-A FUNGICIDES SANKYO COMPANY LIMITED (JP) 1983-12-20 US disclosed
US-4375474-A BACTERICIDES, FUNGICIDES SYNTEX (U.S.A.) INC. (US) 1983-03-01 US disclosed
EP-0055059-A1 Diazole and triazole derivatives, processes for their preparation and anti-microbial compositions containing them SANKYO COMPANY LIMITED (JP) 1982-06-30 EP disclosed
US-4272545-A FUNGICIDES, BACTERICIDE, ANTIPROTOZOA, SPERMATOCIDE SYNTEX (U.S.A.) INC. (US) 1981-06-09 US disclosed
US-4213991-A BACTERICIDES, FUNGICIDES, ANTIPROTOZOA SYNTEX (U.S.A.) INC. (US) 1980-07-22 US disclosed
EP-0005980-A2 Derivatives of substituted N-alkyl imidazoles, their preparation and these compounds for pharmaceutical use SYNTEX (U.S.A.) INC. (US) 1979-12-12 EP disclosed