SCHEMBL4101320

SCHEMBL4101320

O=C(O)N[C@@H]1CCN(C(=O)C(c2cccc(C(F)(F)F)c2)C2CCCCC2)C1

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CHRM3 P20309 4/20 0.45
TEAD1 P28347 2/20 0.44
EPHX2 P34913 3/20 0.44
EPHX1 P07099 1/20 0.44
KLRK1 P26718 1/20 0.43
MICA Q29983 1/20 0.43
LMNA P02545 3/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
GAA P10253 1/20 0.42
MAPT P10636 2/20 0.41
ALOX12 P18054 1/20 0.41
HTT P42858 1/20 0.41
SLC6A9 P48067 1/20 0.41
C3AR1 Q16581 1/20 0.41
ALDH1A1 P00352 1/20 0.41
HTR1E P28566 1/20 0.41
S1PR3 Q99500 1/20 0.41
SIGMAR1 Q99720 1/20 0.41
CNR1 P21554 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4847465 0.85 CHRM3 (0.43) CHRM3EPHX2EPHX1C3AR1
SCHEMBL4955085 0.85 CHRM3 (0.43) CHRM3EPHX2EPHX1C3AR1
SCHEMBL4758293 0.84 CHRM3 (0.47) CHRM3C3AR1CNR1
SCHEMBL3960883 0.84 SLC6A2 (0.45) TEAD1EPHX2EPHX1KLRK1MICA
SCHEMBL3954625 0.84 SLC6A2 (0.45) TEAD1EPHX2EPHX1KLRK1MICA
SCHEMBL4847784 0.81 CHRM3 (0.42) CHRM3EPHX2EPHX1
SCHEMBL4117389 0.81 CHRM3 (0.42) CHRM3EPHX2EPHX1
SCHEMBL3986502 0.78 CHRM3 (0.52) CHRM3EPHX2EPHX1LMNAC3AR1
SCHEMBL3992224 0.78 CHRM3 (0.52) CHRM3EPHX2EPHX1LMNAC3AR1
SCHEMBL3954725 0.77 SLC6A2 (0.46) EPHX2KLRK1MICALMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7550485-B2 Substituted N-heterocycle derivatives and methods of their use WYETH (US) 2009-06-23 US disclosed