SCHEMBL4847784

SCHEMBL4847784

O=C(O)N[C@@H]1CCCN(C(=O)C(c2cccc(OC(F)(F)F)c2)C2CCCCC2)C1

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CHRM3 P20309 4/20 0.42
NOTUM Q6P988 1/20 0.41
MCHR1 Q99705 1/20 0.41
BTK Q06187 2/20 0.40
EPHX1 P07099 2/20 0.40
TAS1R3 Q7RTX0 1/20 0.40
TAS1R1 Q7RTX1 1/20 0.40
TAS1R2 Q8TE23 1/20 0.40
CASR P41180 4/20 0.40
EPHX2 P34913 2/20 0.39
GLS O94925 2/20 0.38
USP30 Q70CQ3 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4117389 1.00 CHRM3 (0.42) CHRM3NOTUMMCHR1BTKEPHX1
SCHEMBL4955085 0.95 CHRM3 (0.43) CHRM3NOTUMEPHX1TAS1R3TAS1R1
SCHEMBL4847465 0.95 CHRM3 (0.43) CHRM3NOTUMEPHX1TAS1R3TAS1R1
SCHEMBL3952527 0.85 SLC6A2 (0.45) NOTUMMCHR1BTKCASR
SCHEMBL3955180 0.85 SLC6A2 (0.45) NOTUMMCHR1BTKCASR
SCHEMBL4565202 0.81 CHRM3 (0.41) CHRM3NOTUMEPHX1USP30
SCHEMBL4101320 0.81 CHRM3 (0.45) CHRM3EPHX1EPHX2
SCHEMBL3961750 0.80 SLC6A2 (0.46) NOTUMEPHX2GLS
SCHEMBL3955877 0.80 SLC6A2 (0.46) NOTUMEPHX2GLS
SCHEMBL1566490 0.78 EPHX1 (0.51) NOTUMEPHX1TAS1R3TAS1R1TAS1R2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7419980-B2 Fused-aryl and heteroaryl derivatives and methods of their use WYETH (US) 2008-09-02 US disclosed
US-7402698-B2 Secondary amino-and cycloamino-cycloalkanol derivatives and methods of their use WYETH (US) 2008-07-22 US disclosed
US-20050234058-A1 Secondary amino-and cycloamino-cycloalkanol derivatives and methods of their use WYETH (US) 2005-10-20 US disclosed
US-20050192283-A1 Fused-aryl and heteroaryl derivatives and methods of their use WYETH (US) 2005-09-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050234058-A1 Secondary amino-and cycloamino-cycloalkanol derivatives and methods of their use ASNS, GLS, GYS1 CHRM3 270/4885NOTUM 1827/4885MCHR1 881/4885
US-20050192283-A1 Fused-aryl and heteroaryl derivatives and methods of their use COMT, MAOA, HTR3A CHRM3 853/4885NOTUM 2347/4885MCHR1 816/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.