SCHEMBL4101464

SCHEMBL4101464

CNC(=O)c1c(-c2ccc(Oc3ccccc3F)cc2)oc2cc(NCS(C)(=O)=O)c(OC)cc12

nearest known ligand 0.41

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
CACNA1C Q13936 1/20 0.39
ANO1 Q5XXA6 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4093302 0.92 CYP2C9 (0.43) CYP3A4CYP2C9CYP2C19CACNA1CANO1
SCHEMBL3395986 0.91 PTGS2 (0.40) CYP3A4CYP2C9CYP2C19CACNA1CANO1
SCHEMBL2842699 0.89 CYP2C9 (0.46) CYP3A4CYP2C9CYP2C19CACNA1CANO1
SCHEMBL16494049 0.88 HPGD (0.39) CYP3A4CYP2C9CYP2C19
SCHEMBL4101460 0.83 CACNA1C (0.50) CACNA1C
SCHEMBL4093610 0.83 CYP3A4 (0.47) CYP3A4CYP2C9CYP2C19CACNA1C
SCHEMBL2842404 0.82 ANO1 (0.54) CYP3A4CYP2C9CYP2C19ANO1
SCHEMBL4094665 0.81 CYP3A4 (0.42) CYP3A4CYP2C9CYP2C19CACNA1CANO1
SCHEMBL3398668 0.81 CYP3A4 (0.46) CYP3A4CYP2C9CYP2C19
SCHEMBL3398507 0.81 CYP2C9 (0.44) CYP3A4CYP2C9CYP2C19CACNA1C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2245023-B1 HETEROCYCLIC ANTIVIRAL COMPOUNDS HOFFMANN LA ROCHE (CH) 2011-12-28 EP claimed
US-8071797-B2 Heterocyclic antiviral compounds ROCHE PALO ALTO LLC (US) 2011-12-06 US claimed
US-20090208449-A1 Heterocyclic antiviral compounds ROCHE PALO ALTO LLC 2009-08-20 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090208449-A1 Heterocyclic antiviral compounds EIF2AK2, HCCS, RTF2 CYP3A4 300/4885CYP2C9 416/4885CYP2C19 594/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.