SCHEMBL411192

SCHEMBL411192

NC(=O)CCc1ccc2ncsc2c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 7/20 0.50
RAB9A P51151 7/20 0.50
TDP1 Q9NUW8 3/20 0.50
KDM4E B2RXH2 3/20 0.50
HKDC1 Q2TB90 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
TGFBR1 P36897 1/20 0.43
SMYD3 Q9H7B4 1/20 0.42
TAS1R3 Q7RTX0 1/20 0.41
TAS1R1 Q7RTX1 1/20 0.41
DYRK1A Q13627 1/20 0.41
GFER P55789 1/20 0.41
ALDH1A1 P00352 2/20 0.40
HTR1A P08908 1/20 0.40
DRD2 P14416 1/20 0.40
HTR2A P28223 1/20 0.40
NAMPT P43490 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL418265 0.86 KDM4E (0.55) NPC1RAB9ATDP1KDM4EHKDC1
SCHEMBL421391 0.84 NPC1 (0.53) NPC1RAB9ATDP1KDM4EHKDC1
SCHEMBL14944865 0.79 DYRK1A (0.46) NPC1RAB9ATDP1KDM4EHKDC1
SCHEMBL5871324 0.79 NPC1 (0.49) NPC1RAB9ATDP1KDM4EHKDC1
Hydrochloric Acid SCHEMBL20562963 0.78 DYRK1A (0.45) NPC1RAB9ATDP1KDM4EHKDC1
SCHEMBL20563305 0.77 NPC1 (0.51) NPC1RAB9ATDP1KDM4EHKDC1
SCHEMBL4943705 0.76 DYRK1A (0.44) NPC1RAB9ATDP1KDM4EHKDC1
SCHEMBL360535 0.76 NPC1 (0.46) NPC1RAB9ATDP1KDM4EHKDC1
SCHEMBL414036 0.76 NPC1 (0.58) NPC1RAB9ATDP1KDM4EHKDC1
SCHEMBL5871480 0.76 NPC1 (0.45) NPC1RAB9ATDP1KDM4EHKDC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103209968-A Pluripotent stem cell cardiomyocyte differentiation-promoting agent UNIV KYOTO 2013-07-17 CN disclosed
EP-2408769-A1 PYRIMIDINE DERIVATIVES USED AS ITK INHIBITORS Glaxo Group Limited (GB) 2012-01-25 EP disclosed
WO-2010106016-A1 PYRIMIDINE DERIVATIVES USED AS ITK INHIBITORS GLAXO GROUP LIMITED (GB) 2010-09-23 WO disclosed