Morpholine

Morpholine

SCHEMBL4121473

C1CCOCC1.C1CCOCC1.C1COCCN1

nearest known ligand 0.94

Full drug profile on Sugi Atlas →

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.69
KMT2A Q03164 1/20 0.69
KDM4E B2RXH2 1/20 0.69
GAA P10253 1/20 0.69
CYP2C9 P11712 1/20 0.69
ALDH1A1 P00352 2/20 0.53
SMN1; SMN2 Q16637 3/20 0.33
APEX1 P27695 1/20 0.33
CXCR4 P61073 1/20 0.33
HTT P42858 1/20 0.33
LMNA P02545 1/20 0.32
TTR P02766 1/20 0.31
HIF1A Q16665 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Morpholine SCHEMBL22582364 1.00 MEN1 (0.69) MEN1KMT2AKDM4EGAACYP2C9
SCHEMBL5314604 0.97 MEN1 (0.75) MEN1KMT2AKDM4EGAACYP2C9
Morpholine SCHEMBL11883179 0.97 MEN1 (0.65) MEN1KMT2AKDM4EGAACYP2C9
SCHEMBL9400799 0.97 MEN1 (0.75) MEN1KMT2AKDM4EGAACYP2C9
Morpholine SCHEMBL1932496 0.97 MEN1 (0.73) MEN1KMT2AKDM4EGAACYP2C9
SCHEMBL622411 0.94 MEN1 (0.61) MEN1KMT2AKDM4EGAACYP2C9
SCHEMBL9400796 0.94 MEN1 (0.71) MEN1KMT2AKDM4EGAACYP2C9
SCHEMBL27478132 0.94 MEN1 (0.61) MEN1KMT2AKDM4EGAACYP2C9
SCHEMBL19992556 0.94 MEN1 (0.61) MEN1KMT2AKDM4EGAACYP2C9
SCHEMBL1824995 0.94

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8318730-B2 Fused hetrocyclic compounds SYNTA PHARMACEUTICALS CORPORATION (US) 2012-11-27 US disclosed
US-7615552-B2 Fused heterocyclic compounds SYNTA PHARMACEUTICALS CORP. (US) 2009-11-10 US disclosed
US-20090253694-A1 Fused hetrocyclic compounds SYNTA PHARMACEUTICALS CORP. (US) 2009-10-08 US disclosed
US-20050250770-A1 Fused heterocyclic compounds LSI FINANCING LLC, AS ADMINISTRATIVE AGENT 2005-11-10 US disclosed
EP-0785765-B1 AGENT AND PROCESS FOR PERMANENTLY SHAPING KERATIN FIBRES HENKEL KGAA (DE) 2002-04-03 EP disclosed
EP-0785765-A1 AGENT AND PROCESS FOR PERMANENTLY SHAPING KERATIN FIBRES Henkel Kommanditgesellschaft auf Aktien (DE) 1997-07-30 EP disclosed
WO-1996010986-A1 AGENT AND PROCESS FOR PERMANENTLY SHAPING KERATIN FIBRES HENKEL KOMMANDITGESELLSCHAFT AUF AKTIEN (DE) 1996-04-18 WO disclosed
US-3989640-A SYNERGISTIC, MORPHOLINE, AMMONIUM BENZOATE AND CYCLOHEXANE OR NITROPROPANE OR CYCLOPENTENE THE DRACKETT COMPANY (US) 1976-11-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050250770-A1 Fused heterocyclic compounds IL2, IL4, IL15 MEN1 1246/4885KMT2A 2143/4885KDM4E 3523/4885
US-20090253694-A1 Fused hetrocyclic compounds IL2, IL15, IL4 MEN1 1345/4885KMT2A 2644/4885KDM4E 3697/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.