SCHEMBL4123057

SCHEMBL4123057

Cc1nc2ccc(F)cc2c(=O)o1

nearest known ligand 0.70

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ELANE P08246 10/20 0.70
CASP3 P42574 1/20 0.49
HPN P05981 1/20 0.45
TYMS P04818 1/20 0.44
MPO P05164 1/20 0.44
IDO1 P14902 1/20 0.42
TDO2 P48775 1/20 0.42
IDO2 Q6ZQW0 1/20 0.42
ALDH1A1 P00352 2/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
KDM4E B2RXH2 1/20 0.41
POLB P06746 1/20 0.41
PTK2B Q14289 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12789755 0.87 ELANE (0.57) ELANECASP3KMT2A
SCHEMBL4113871 0.86 ELANE (0.59) ELANECASP3TYMSMPOALDH1A1
SCHEMBL30089873 0.86 ELANE (0.59) ELANECASP3TYMSMPOALDH1A1
SCHEMBL12789630 0.82 ELANE (0.56) ELANECASP3HPNIDO1TDO2
SCHEMBL4117968 0.82 ELANE (1.00) ELANEALDH1A1MEN1KMT2AKDM4E
SCHEMBL3539033 0.79 ELANE (0.70) ELANETYMSALDH1A1MEN1KMT2A
SCHEMBL12847193 0.79 ELANE (0.70) ELANEALDH1A1MEN1KMT2AKDM4E
SCHEMBL12352004 0.79 ELANE (0.70) ELANEMEN1KMT2A
SCHEMBL1812732 0.79 ELANE (0.70) ELANETYMSMPOALDH1A1MEN1
SCHEMBL12758386 0.79 ELANE (0.70) ELANEALDH1A1MEN1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119954731-A Chalcone derivative containing 4-quinazolinone structure, and preparation method and application thereof 黔南州烟草公司平塘县分公司 2025-05-09 CN disclosed
CN-115677803-B Preparation method of glycoside derivative containing quinazoline structure and composition thereof and application of glycoside derivative and composition for preventing and treating kiwi fruit canker 贵州理工学院 2025-03-28 CN disclosed
CN-115521261-B Preparation method of mercapto-containing quinazolinone and composition thereof, and application of mercapto-containing quinazolinone in resisting kiwi fruit canker 贵州理工学院 2024-04-05 CN disclosed
CN-115636795-B Preparation method of quinazolinone derivative containing thiobenzamide structure and composition thereof, and application of quinazolinone derivative and composition thereof in preventing and treating kiwi fruit canker 贵州理工学院 2024-04-05 CN disclosed
CN-115521262-B Preparation method of quinazolinone containing phenyl and composition thereof, and application of quinazolinone and composition in resisting kiwi fruit canker 贵州理工学院 2024-04-05 CN disclosed
CN-115677803-A Preparation method of glucoside derivative containing quinazoline structure, preparation method of composition of glucoside derivative and application of composition in prevention and treatment of kiwifruit canker 贵州理工学院 2023-02-03 CN disclosed
CN-115636795-A Quinazolinone derivative containing thiobenzamide structure, composition and application of quinazolinone derivative in prevention and treatment of kiwifruit canker 贵州理工学院 2023-01-24 CN disclosed
CN-115521261-A Preparation method of sulfhydryl-containing quinazolinone and composition thereof and application of sulfhydryl-containing quinazolinone in resisting kiwifruit canker 贵州理工学院 2022-12-27 CN disclosed
CN-115521262-A Preparation method of phenyl-containing quinazolinone and composition thereof and application of phenyl-containing quinazolinone in resisting kiwifruit canker 贵州理工学院 2022-12-27 CN disclosed
US-20090181942-A1 TRICYCLIC COMPOUNDS DAIICHI SANKYO COMPANY, LIMITED (JP) 2009-07-16 US disclosed
EP-1939205-A1 TRICYCLIC COMPOUND Daiichi Sankyo Company, Limited (JP) 2008-07-02 EP disclosed
EP-0552665-A1 Pyrrolylbenzodiazepinones and medicines containing them F. HOFFMANN-LA ROCHE AG (CH) 1993-07-28 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090181942-A1 TRICYCLIC COMPOUNDS FDFT1, COASY, HMGCR ELANE 2050/4885CASP3 3424/4885HPN 223/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.