SCHEMBL4123352

SCHEMBL4123352

Cc1ccc(NC(=O)Nc2cccc(-c3ccnc(C)n3)c2)cc1

nearest known ligand 0.82

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.82
CNR1 P21554 10/20 0.62
KDR P35968 2/20 0.54
NPC1 O15118 1/20 0.52
RAB9A P51151 1/20 0.52
CNR2 P34972 1/20 0.52
FGFR3 P22607 1/20 0.52
PLK1 P53350 1/20 0.51
DNMT3B Q9UBC3 2/20 0.51
EPHB4 P54760 1/20 0.50
RAF1 P04049 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4921357 0.92 MAPT (0.82) MAPTCNR1KDRRAB9ACNR2
SCHEMBL4118606 0.91 MAPT (0.76) MAPTCNR1KDRNPC1RAB9A
SCHEMBL4922831 0.90 MAPT (0.79) MAPTCNR1KDRNPC1RAB9A
SCHEMBL4912509 0.90 MAPT (1.00) MAPTCNR1CNR2
Hydrochloric Acid SCHEMBL4915559 0.89 MAPT (0.98) MAPTCNR1CNR2
SCHEMBL4915532 0.84 MAPT (0.70) MAPTCNR1NPC1RAB9ADNMT3B
SCHEMBL4119185 0.84 MAPT (0.70) MAPTCNR1KDRCNR2FGFR3
SCHEMBL4922785 0.78 MAPT (0.61) MAPTCNR1
SCHEMBL8312358 0.77 PLK1 (0.59) MAPTKDRFGFR3PLK1DNMT3B
SCHEMBL20557632 0.77 CNR1 (1.00) MAPTCNR1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1804785-A2 DIARYL UREAS AS CB1 ANTAGONISTS NEUROGEN CORPORATION (US) 2007-07-11 EP claimed
WO-2006049941-A2 DIARYL UREAS AS CB1 ANTAGONISTS NEUROGEN CORPORATION (US) 2006-05-11 WO claimed
US-20090239841-A1 Diaryl Ureas as CB1 Antagonists NEUROGEN CORPORATION 2009-09-24 US disclosed
US-20090239841-A1 Diaryl Ureas as CB1 Antagonists NEUROGEN CORPORATION 2009-09-24 US disclosed
US-20090239841-A1 Diaryl Ureas as CB1 Antagonists NEUROGEN CORPORATION 2009-09-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090239841-A1 Diaryl Ureas as CB1 Antagonists CNR1, CNR2, OPRL1 MAPT 1654/4885CNR1 1/4885KDR 3246/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.