SCHEMBL4124748

SCHEMBL4124748

CN(NC(=O)c1c(NS(C)(=O)=O)nn2c(-c3ccc(Cl)cc3)c(-c3ccccc3Cl)cnc12)c1ccccn1

nearest known ligand 0.34

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 10/20 0.34
MAPT P10636 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
MAPK10 P53779 2/20 0.33
GLO1 Q04760 1/20 0.32
TDP1 Q9NUW8 1/20 0.31
MAP4K4 O95819 1/20 0.30
LMNA P02545 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4124736 0.89 CNR1 (0.34) CNR1MAPTSMN1; SMN2TDP1
SCHEMBL2086773 0.88 F10 (0.34) CNR1MAPTSMN1; SMN2TDP1
SCHEMBL2085682 0.88 CNR1 (0.33) CNR1MAPTSMN1; SMN2TDP1LMNA
SCHEMBL2085825 0.87 MAPT (0.32) CNR1MAPTSMN1; SMN2TDP1LMNA
SCHEMBL4121879 0.85 HTT (0.36) CNR1MAPTSMN1; SMN2TDP1LMNA
SCHEMBL4121872 0.84 MAP4K4 (0.36) CNR1MAPTSMN1; SMN2MAP4K4
SCHEMBL4112770 0.84 NPC1 (0.33) CNR1MAPTSMN1; SMN2TDP1LMNA
SCHEMBL2084584 0.84 MALT1 (0.32) CNR1MAPTSMN1; SMN2
SCHEMBL2083247 0.83 CNR1 (0.40) CNR1
SCHEMBL4121225 0.81 JAK2 (0.36) MAPTSMN1; SMN2TDP1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8188097-B2 Pyrazolo[1,5-A]pyrimidine compounds MITSUBISHI TANABE PHARMA CORPORATION (JP) 2012-05-29 US disclosed
US-20090069298-A1 Pyrazolo[1,5-A]Pyrimidine Compounds TANABE SEIYAKU CO., LTD. (JP) 2009-03-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090069298-A1 Pyrazolo[1,5-A]Pyrimidine Compounds RECQL, QTRT1, DPYD CNR1 285/4885MAPT 4568/4885SMN1; SMN2 3307/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.