SCHEMBL4128470

SCHEMBL4128470

Cc1ccc(NC(=O)c2cccc(C(F)(F)F)c2)cc1NC(=O)Nc1ccc2c(c1)NC(=O)C2=Cc1[nH]c(C)c(C(=O)O)c1C

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FLT3 P36888 9/20 0.65
FLT4 P35916 5/20 0.65
KDR P35968 5/20 0.65
KIT P10721 3/20 0.65
NTRK1 P04629 4/20 0.62
AURKB Q96GD4 5/20 0.57
CSF1R P07333 6/20 0.56
NTRK3 Q16288 2/20 0.53
MET P08581 2/20 0.52
PDGFRB P09619 2/20 0.52
AURKA O14965 1/20 0.52
AURKC Q9UQB9 1/20 0.52
NTRK2 Q16620 2/20 0.52
JAK2 O60674 1/20 0.52
ABL1 P00519 1/20 0.52
INSR P06213 1/20 0.52
LYN P07948 1/20 0.52
RET P07949 1/20 0.52
IGF1R P08069 1/20 0.52
ROS1 P08922 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4128467 1.00 FLT3 (0.65) FLT3FLT4KDRKITNTRK1
SCHEMBL5007514 0.94 NTRK1 (0.66) FLT3FLT4KDRKITNTRK1
SCHEMBL5007515 0.94 NTRK1 (0.66) FLT3FLT4KDRKITNTRK1
SCHEMBL396702 0.93 NTRK1 (0.69) FLT3FLT4KDRKITNTRK1
SCHEMBL396701 0.93 NTRK1 (0.69) FLT3FLT4KDRKITNTRK1
SCHEMBL4133365 0.90 FLT3 (0.77) FLT3FLT4KDRKITNTRK1
SCHEMBL4133367 0.90 FLT3 (0.77) FLT3FLT4KDRKITNTRK1
SCHEMBL4122462 0.89 NTRK1 (0.76) FLT3FLT4KDRKITNTRK1
SCHEMBL3997804 0.89 NTRK1 (0.76) FLT3FLT4KDRKITNTRK1
SCHEMBL10091879 0.87 FLT3 (0.60) FLT3FLT4KDRKITNTRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1814545-A4 COMPOUNDS AND COMPOSITIONS AS PROTEIN KINASE INHIBITORS IRM LLC (BM) 2009-06-10 EP claimed
US-20080221192-A1 Compounds and Compositions as Protein Kinase Inhibitors IRM LLC (BM) 2008-09-11 US claimed
EP-1814545-A2 COMPOUNDS AND COMPOSITIONS AS PROTEIN KINASE INHIBITORS IRM, LLC (BM) 2007-08-08 EP claimed
WO-2006052936-A2 COMPOUNDS AND COMPOSITIONS AS PROTEIN KINASE INHIBITORS IRM LLC (BM) 2006-05-18 WO claimed
EP-1814545-A4 COMPOUNDS AND COMPOSITIONS AS PROTEIN KINASE INHIBITORS IRM LLC (BM) 2009-06-10 EP disclosed
US-20080221192-A1 Compounds and Compositions as Protein Kinase Inhibitors IRM LLC (BM) 2008-09-11 US disclosed
EP-1814545-A2 COMPOUNDS AND COMPOSITIONS AS PROTEIN KINASE INHIBITORS IRM, LLC (BM) 2007-08-08 EP disclosed
WO-2006052936-A2 COMPOUNDS AND COMPOSITIONS AS PROTEIN KINASE INHIBITORS IRM LLC (BM) 2006-05-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080221192-A1 Compounds and Compositions as Protein Kinase Inhibitors BMX, FRK, PTK2B FLT3 93/4885FLT4 323/4885KDR 204/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.