SCHEMBL41315

SCHEMBL41315

Oc1ccc(Cl)c(-c2ccc3nc(Nc4cccc(C(O)O)c4)ncc3c2)c1

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAP3K5 Q99683 3/20 0.42
ABL1 P00519 2/20 0.42
PDGFRB P09619 3/20 0.41
SRC P12931 3/20 0.41
SYK P43405 4/20 0.40
BRAF P15056 5/20 0.40
LCK P06239 1/20 0.40
EGFR P00533 1/20 0.39
FGFR1 P11362 1/20 0.39
PDGFRA P16234 1/20 0.39
MAPK14 Q16539 1/20 0.39
YES1 P07947 1/20 0.39
EPHB4 P54760 1/20 0.39
FGFR4 P22455 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL42236 0.83 SRC (0.57) MAP3K5ABL1PDGFRBSRCBRAF
SCHEMBL42013 0.79 BRAF (0.43) MAP3K5ABL1PDGFRBSRCSYK
SCHEMBL41314 0.78 BRAF (0.42) ABL1PDGFRBSRCBRAFEGFR
SCHEMBL40934 0.77 SYK (0.47) MAP3K5ABL1SRCSYKBRAF
SCHEMBL41349 0.76 SRC (0.62) PDGFRBSRCBRAFEGFRFGFR1
SCHEMBL42217 0.76 JAK2 (0.47) SRCBRAFLCKEGFRFGFR1
SCHEMBL42295 0.76 BRAF (0.43) ABL1PDGFRBSRCBRAF
SCHEMBL41009 0.75 LRRK2 (0.47) PDGFRBSRC
SCHEMBL41686 0.75 SRC (0.39) ABL1PDGFRBSRCYES1
SCHEMBL40938 0.73 SRC (0.40) ABL1PDGFRBSRCBRAFLCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20130123271-A1 HETEROCYCLIC COMPOUNDS, THEIR PREPARATION AND THERAPEUTIC APPLICATION FOVEA PHARMACEUTICALS (FR) 2013-05-16 US claimed
EP-2585439-A1 HETEROCYCLIC COMPOUNDS, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION Fovea Pharmaceuticals (FR) 2013-05-01 EP claimed
WO-2011161159-A1 HETEROCYCLIC COMPOUNDS, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION FOVEA PHARMACEUTICALS (FR) 2011-12-29 WO claimed
US-20130123271-A1 HETEROCYCLIC COMPOUNDS, THEIR PREPARATION AND THERAPEUTIC APPLICATION FOVEA PHARMACEUTICALS (FR) 2013-05-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130123271-A1 HETEROCYCLIC COMPOUNDS, THEIR PREPARATION AND THERAPEUTIC APPLICATION CAMK2D, CAMK2A, CAMK2B MAP3K5 145/4885ABL1 181/4885PDGFRB 803/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.