Epoprostenol

Epoprostenol

SCHEMBL41345

CCCCC[C@H](O)C=C[C@@H]1[C@H]2CC(=CCCCC(=O)O)O[C@H]2C[C@H]1O.[NaH]

nearest known ligand 0.98

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

PTGIR

The experimentally established mechanism targets of Epoprostenol. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGIR known ✓ P43119 6/20 0.55
ALDH1A1 P00352 5/20 0.98
MEN1 O00255 2/20 0.70
KMT2A Q03164 2/20 0.70
PPARG P37231 1/20 0.70
PPARD Q03181 1/20 0.70
PPARA Q07869 1/20 0.70
PTGER4 P35408 4/20 0.56
TBXA2R P21731 3/20 0.56
LMNA P02545 3/20 0.56
PTGER1 P34995 2/20 0.56
PTGFR P43088 2/20 0.56
PTGER3 P43115 2/20 0.56
PTGDR Q13258 1/20 0.56
SLCO2A1 Q92959 1/20 0.56
PTGER2 P43116 3/20 0.55
TSHR P16473 3/20 0.55
HPGD P15428 3/20 0.55
MAPK1 P28482 2/20 0.55
NR1I2 O75469 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Epoprostenol SCHEMBL2821707 1.00 ALDH1A1 (0.98) ALDH1A1MEN1KMT2APPARGPPARD
Epoprostenol SCHEMBL705594 0.99 ALDH1A1 (1.00) ALDH1A1MEN1KMT2APPARGPPARD
Epoprostenol SCHEMBL22607961 0.99 ALDH1A1 (1.00) ALDH1A1MEN1KMT2APPARGPPARD
Epoprostenol SCHEMBL551616 0.99 ALDH1A1 (1.00) ALDH1A1MEN1KMT2APPARGPPARD
Epoprostenol SCHEMBL24612535 0.99 ALDH1A1 (1.00) ALDH1A1MEN1KMT2APPARGPPARD
Epoprostenol SCHEMBL24033081 0.99 ALDH1A1 (1.00) ALDH1A1MEN1KMT2APPARGPPARD
Epoprostenol SCHEMBL4165739 0.99 ALDH1A1 (1.00) ALDH1A1MEN1KMT2APPARGPPARD
Epoprostenol SCHEMBL24340812 0.99 ALDH1A1 (1.00) ALDH1A1MEN1KMT2APPARGPPARD
Epoprostenol SCHEMBL21283002 0.99 ALDH1A1 (1.00) ALDH1A1MEN1KMT2APPARGPPARD
Epoprostenol SCHEMBL16783375 0.99 ALDH1A1 (1.00) ALDH1A1MEN1KMT2APPARGPPARD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1399 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240282425-A1 AUTHENTICATION METHODS AND SYSTEMS FOR DISPENSED PRESCRIPTIONS LOW GORDON KEITH (US) 2024-08-22 US claimed
CN-117887421-A Ultrahigh-heat-conductivity graphene foam energy storage material and preparation method thereof 中国空间技术研究院 2024-04-16 CN claimed
EP-4069826-A1 EXTRACELLULAR VESICLES AND THEIR USES United Therapeutics Corporation (US) 2022-10-12 EP claimed
CN-109153660-B Method for preparing epoprostenol sodium with enhanced stability 奇诺因药物和化学工厂私人有限公司 2022-10-11 CN claimed
CN-115066491-A Extracellular vesicles and uses thereof 联合治疗公司 2022-09-16 CN claimed
US-20220211645-A1 Maximizing Distribution and Minimizing Washout of Injectates in Bone and Method for Enhanced Aspirate Extraction YALE UNIVERSITY 2022-07-07 US claimed
EP-3965635-A2 MAXIMIZING DISTRIBUTION AND MINIMIZING WASHOUT OF INJECTATES IN BONE AND METHOD FOR ENHANCED ASPIRATE EXTRACTION Yale University (US) 2022-03-16 EP claimed
EP-3852608-A1 COMPOSITIONS AND METHODS FOR GLAUCOMA Aufbau Medical Innovations Limited (IE) 2021-07-28 EP claimed
WO-2021113299-A1 EXTRACELLULAR VESICLES AND THEIR USES UNITED THERAPEUTICS CORPORATION (US) 2021-06-10 WO claimed
CN-107921202-B Reducing leakage during refilling of implantable injection devices 美敦力公司 2021-06-04 CN claimed
WO-2002026318-A1 METHOD AND SYSTEM FOR NERVE STIMULATION AND CARDIAC SENSING PRIOR TO AND DURING A MEDICAL PROCEDURE MEDTRONIC, INC. (US) 2002-04-04 WO claimed
US-4430340-A HEXADECYLTRIMETHYLAMMONIUM CHLORIDE, WATER, PROSTACYCLIN SODIUM SALT, DRUGS THE UPJOHN COMPANY (US) 1984-02-07 US claimed
US-4404212-A ADMINISTERING ALONG WITH A HYDROLASE INHIBITOR; ANTICOAGULANTS BURROUGHS WELLCOME CO. (US) 1983-09-13 US claimed
EP-0005768-B1 PHARMACEUTICAL FORMULATIONS CONTAINING PROSTAGLANDIN COMPOUNDS AND METHOD FOR THEIR PREPARATION THE WELLCOME FOUNDATION LIMITED (GB) 1983-08-10 EP claimed
US-4393063-A SYNERGISTIC COMBINATION OF LA PROSTACYCLINE AND A PHOSPHODIESTERASE INHIBITOR BURROUGHS WELLCOME CO. (US) 1983-07-12 US claimed
EP-0007245-B1 PHARMACEUTICAL COMPOSITIONS COMPRISING PROSTACYCLIN OR A PROSTACYCLIN ANALOGUE CONTAINING AN ENOL ETHER GROUP THE UPJOHN COMPANY (US) 1982-12-08 EP claimed
US-4337254-A ANTICOAGULANTS COMPRISING A PROSTACYCLIN AND A PHOSPHODIESTERASE INHIBITOR; PREVENTING LOWERING OF BLOOD PRESSURE BURROUGHS WELLCOME CO. (US) 1982-06-29 US claimed
US-4335139-A PROSTAGLANDINS BURROUGHS WELLCOME CO. (US) 1982-06-15 US claimed
EP-0007245-A1 Pharmaceutical compositions comprising prostacyclin or a prostacyclin analogue containing an enol ether group THE UPJOHN COMPANY (US) 1980-01-23 EP claimed
EP-0005768-A1 Pharmaceutical formulations containing prostaglandin compounds and method for their preparation THE WELLCOME FOUNDATION LIMITED (GB) 1979-12-12 EP claimed