SCHEMBL4135581

SCHEMBL4135581

O=CCc1ccc(-c2cnc(N3CCC4(CC3)CCN(C3CCC3)CC4)nc2)cc1

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TLR9 Q9NR96 3/20 0.38
TLR8 Q9NR97 3/20 0.38
TLR7 Q9NYK1 3/20 0.38
TLR4 O00206 1/20 0.37
HRH3 Q9Y5N1 8/20 0.37
AOC3 Q16853 1/20 0.35
FFAR4 Q5NUL3 1/20 0.35
KDM2B Q8NHM5 1/20 0.34
ACHE P22303 1/20 0.34
POLB P06746 1/20 0.34
KCNH2 Q12809 1/20 0.33
ADRA1A P35348 1/20 0.33
CHRM1 P11229 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4141352 0.85 FFAR4 (0.48) HRH3FFAR4
SCHEMBL14027061 0.82 RET (0.41) TLR9TLR8TLR7
SCHEMBL4130708 0.82 HRH3 (0.43) TLR9TLR8TLR7TLR4HRH3
SCHEMBL4136516 0.81 HRH3 (0.47) HRH3FFAR4
SCHEMBL4935121 0.80 HRH3 (0.41) TLR9TLR8TLR7TLR4HRH3
SCHEMBL4136337 0.79 HRH3 (0.44) TLR9TLR8TLR7TLR4HRH3
SCHEMBL4928014 0.79 HRH3 (0.46) TLR9TLR8TLR7HRH3ADRA1A
SCHEMBL4140025 0.79 SCD (0.40) HRH3
SCHEMBL4131497 0.78 HRH3 (0.44) TLR9TLR8TLR7HRH3KDM2B
SCHEMBL1744283 0.76 TLR9 (0.42) TLR9TLR8TLR7TLR4HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2021004-A2 SUBSTITUTED AZASPIRO DERIVATIVES NEUROGEN CORPORATION (US) 2009-02-11 EP disclosed
WO-2007133561-A2 SUBSTITUTED AZASPIRO DERIVATIVES NEUROGEN CORPORATION (US) 2007-11-22 WO disclosed