SCHEMBL4138243

SCHEMBL4138243

Cn1c(=O)[nH]c(N2CCN(Cc3ccccc3)CC2)c(Cc2ccccc2)c1=O

nearest known ligand 0.77

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 11/20 0.77
ALDH1A1 P00352 3/20 0.49
GLA P06280 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
MAPK1 P28482 2/20 0.48
HTT P42858 2/20 0.48
POLB P06746 1/20 0.47
MC4R P32245 1/20 0.47
TSHR P16473 2/20 0.46
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4151371 0.87 NR3C1 (1.00) NR3C1HTT
SCHEMBL4138311 0.82 NR3C1 (0.72) NR3C1MEN1KMT2A
SCHEMBL4147688 0.81 NR3C1 (1.00) NR3C1ALDH1A1MAPK1HTTMEN1
SCHEMBL4151366 0.81 NR3C1 (1.00) NR3C1
SCHEMBL4138314 0.80 NR3C1 (0.66) NR3C1MAPK1TSHRMEN1KMT2A
SCHEMBL4143729 0.79 NR3C1 (1.00) NR3C1ALDH1A1HTT
SCHEMBL4151367 0.79 NR3C1 (1.00) NR3C1ALDH1A1
SCHEMBL4142930 0.78 NR3C1 (1.00) NR3C1
SCHEMBL4151237 0.76 NR3C1 (0.89) NR3C1ALDH1A1MAPK1HTTMEN1
SCHEMBL2672956 0.76 NR3C1 (0.59) NR3C1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8173664-B2 Modified pyrimidine glucocorticoid receptor modulators CORCEPT THERAPEUTICS, INC. (US) 2012-05-08 US disclosed
US-8173664-B2 Modified pyrimidine glucocorticoid receptor modulators CORCEPT THERAPEUTICS, INC. (US) 2012-05-08 US disclosed
US-7576076-B2 Modified pyrimidine glucocorticoid receptor modulators CORCEPT THERAPEUTICS, INC. (US) 2009-08-18 US disclosed
US-7576076-B2 Modified pyrimidine glucocorticoid receptor modulators CORCEPT THERAPEUTICS, INC. (US) 2009-08-18 US disclosed