SCHEMBL4147298

SCHEMBL4147298

C=CC1CCCN(C(=O)OC(C)(C)C)C1

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.51
ALDH1A1 P00352 1/20 0.51
MAPT P10636 1/20 0.51
KMT2A Q03164 1/20 0.51
HPGD P15428 1/20 0.49
EPHX1 P07099 1/20 0.43
PREP P48147 2/20 0.42
USP2 O75604 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
USP30 Q70CQ3 1/20 0.41
RECQL P46063 1/20 0.40
HSD17B10 Q99714 1/20 0.40
NR1H2 P55055 1/20 0.40
GLS O94925 2/20 0.40
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
HPGDS O60760 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22731686 1.00 MEN1 (0.51) MEN1ALDH1A1MAPTKMT2AHPGD
SCHEMBL25467053 1.00 MEN1 (0.51) MEN1ALDH1A1MAPTKMT2AHPGD
SCHEMBL1279722 0.91 HPGD (0.48) MEN1ALDH1A1MAPTKMT2AHPGD
SCHEMBL344569 0.91 HPGD (0.48) MEN1ALDH1A1MAPTKMT2AHPGD
SCHEMBL344797 0.91 HPGD (0.48) MEN1ALDH1A1MAPTKMT2AHPGD
SCHEMBL1992277 0.86 MEN1 (0.52) MEN1ALDH1A1MAPTKMT2AHPGD
SCHEMBL192730 0.86 MEN1 (0.52) MEN1ALDH1A1MAPTKMT2AHPGD
SCHEMBL641613 0.86 MEN1 (0.52) MEN1ALDH1A1MAPTKMT2AHPGD
SCHEMBL23034653 0.85 MEN1 (0.51) MEN1ALDH1A1MAPTKMT2AHPGD
SCHEMBL6915624 0.84 NR1H2 (0.50) MEN1ALDH1A1MAPTKMT2AHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025026392-A1 KINESIN KIF18A INHIBITOR AND USE THEREOF 上海湃隆生物科技有限公司 2025-02-06 WO disclosed
CN-114502540-A TEAD inhibitors and uses thereof 医肯纳肿瘤学公司 2022-05-13 CN disclosed
EP-3889154-A1 HETEROCYCLIC COMPOUND INTERMEDIATE, PREPARATION METHOD THEREFOR AND APPLICATION THEREOF Wuhan LL Science And Technology Development Co., Ltd. (CN) 2021-10-06 EP disclosed
EP-2683716-A1 PYRIDO[3,4-B]PYRAZINE DERIVATIVES AS SYK INHIBITORS Glaxo Group Limited (GB) 2014-01-15 EP disclosed
US-20140005188-A1 PYRIDO[3,4-B]PYRAZINE DERIVATIVES AS SYK INHIBITORS GLAXO GROUP LIMITED (GB) 2014-01-02 US disclosed
WO-2012123312-A1 PYRIDO[3,4-B]PYRAZINE DERIVATIVES AS SYK INHIBITORS GLAXO GROUP LIMITED (GB) 2012-09-20 WO disclosed
WO-2012123312-A1 PYRIDO[3,4-B]PYRAZINE DERIVATIVES AS SYK INHIBITORS GLAXO GROUP LIMITED (GB) 2012-09-20 WO disclosed
US-20090192169-A1 Bicyclic Benzimidazole Compounds and Their Use as Metabotropic Glutamate Receptor Potentiators ASTRAZENECA AB (SE) 2009-07-30 US disclosed
US-20090192169-A1 Bicyclic Benzimidazole Compounds and Their Use as Metabotropic Glutamate Receptor Potentiators ASTRAZENECA AB (SE) 2009-07-30 US disclosed
US-20090192169-A1 Bicyclic Benzimidazole Compounds and Their Use as Metabotropic Glutamate Receptor Potentiators ASTRAZENECA AB (SE) 2009-07-30 US disclosed
WO-2007115077-A2 BICYCLIC BENZIMIDAZOLE COMPOUNDS AND THEIR USE AS METABOTROPIC GLUTAMATE RECEPTOR POTENTIATORS ASTRAZENECA AB (SE) 2007-10-11 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140005188-A1 PYRIDO[3,4-B]PYRAZINE DERIVATIVES AS SYK INHIBITORS SYK, BTK, LCK MEN1 3382/4885ALDH1A1 2833/4885MAPT 3206/4885
US-20090192169-A1 Bicyclic Benzimidazole Compounds and Their Use as Metabotropic Glutamate Receptor Potentiators GRM1, GRIN1, GRM2 MEN1 3345/4885ALDH1A1 1006/4885MAPT 3505/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.