SCHEMBL4148741

SCHEMBL4148741

O=C(O)c1ccc2cc3n(c2c1)/C=C\N=C/c1ccccc1-3

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.38
POLB P06746 1/20 0.38
ALDH1A1 P00352 2/20 0.36
KDM4E B2RXH2 1/20 0.36
HPGD P15428 1/20 0.36
ACLY P53396 2/20 0.35
TTR P02766 1/20 0.35
FGFR1 P11362 1/20 0.34
NR1H2 P55055 1/20 0.34
NR1H3 Q13133 1/20 0.34
PTPRC P08575 2/20 0.34
MEN1 O00255 1/20 0.34
PKM P14618 1/20 0.34
HTT P42858 1/20 0.34
RAB9A P51151 1/20 0.34
RXFP1 Q9HBX9 1/20 0.34
AURKA O14965 1/20 0.34
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3092075 0.79 SRPK1 (0.34) ACLY
SCHEMBL3244153 0.74 SRD5A2 (0.43) KMT2APOLBALDH1A1KDM4EHPGD
SCHEMBL4139797 0.73 KMT2A (0.37) KMT2APOLBALDH1A1KDM4EHPGD
SCHEMBL3075059 0.71 TBXA2R (0.36) KMT2APOLBALDH1A1KDM4EHPGD
SCHEMBL4823474 0.70 POLB (0.36) KMT2APOLBKDM4EACLYFGFR1
SCHEMBL3236134 0.69 KMT2A (0.38) KMT2APOLBALDH1A1KDM4EHPGD
SCHEMBL270972 0.68 POLB (0.40) KMT2APOLBALDH1A1KDM4EHPGD
SCHEMBL3943354 0.68 SRD5A2 (0.48) KMT2APOLBALDH1A1KDM4EHPGD
SCHEMBL50870 0.68 POLB (0.39) KMT2APOLBALDH1A1KDM4EHPGD
SCHEMBL4830030 0.66 SLC22A12 (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090136449-A1 Tetracyclic Indole Derivatives as Antiviral Agents ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI SPA (IT) 2009-05-28 US claimed
US-20090136449-A1 Tetracyclic Indole Derivatives as Antiviral Agents ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI SPA (IT) 2009-05-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090136449-A1 Tetracyclic Indole Derivatives as Antiviral Agents IDO1, IDO2, ZC3HAV1 KMT2A 3385/4885POLB 4396/4885ALDH1A1 754/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.