SCHEMBL3092075

SCHEMBL3092075

O=C(O)c1ccc2cc3n(c2c1)/C=C\N=C/c1ccsc1-3

nearest known ligand 0.34

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SRPK1 Q96SB4 1/20 0.34
RPS6KB2 Q9UBS0 1/20 0.34
AKR1C3 P42330 1/20 0.31
MAPKAPK2 P49137 3/20 0.31
CSNK2A2 P19784 1/20 0.30
CSNK2B P67870 1/20 0.30
CSNK2A1 P68400 1/20 0.30
RPS6KA3 P51812 1/20 0.30
ACLY P53396 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4148741 0.79 KMT2A (0.38) ACLY
SCHEMBL4148744 0.79 KMT2A (0.38) ACLY
SCHEMBL4830100 0.64 KDM4E (0.37) SRPK1RPS6KB2MAPKAPK2CSNK2A1RPS6KA3
SCHEMBL4826413 0.63 MAPK8 (0.34) MAPKAPK2RPS6KA3
SCHEMBL4825624 0.61 CA12 (0.35) SRPK1RPS6KB2RPS6KA3ACLY
SCHEMBL3244153 0.60 SRD5A2 (0.43) AKR1C3ACLY
SCHEMBL4830030 0.60 SLC22A12 (0.35) MAPKAPK2CSNK2A2CSNK2BCSNK2A1RPS6KA3
SCHEMBL4139797 0.60 KMT2A (0.37) ACLY
SCHEMBL3236134 0.58 KMT2A (0.38) ACLY
SCHEMBL17515229 0.58 TDP1 (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7795247-B2 Tetracyclic indole derivatives as antiviral agents ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI SPA (IT) 2010-09-14 US disclosed
US-20060100262-A1 Tetracyclic indole derivatives as antiviral agents ISTITUTO DI RICHERCHEDI BIOLOGIA MOLECOLARE P ANGELETTI SPA (IRMB) (IT) 2006-05-11 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060100262-A1 Tetracyclic indole derivatives as antiviral agents IDO1, ZC3HAV1, IDO2 SRPK1 2862/4885RPS6KB2 3519/4885AKR1C3 241/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.