SCHEMBL4153461

SCHEMBL4153461

COc1cc2c(=O)[nH]cnc2cc1C(=O)O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRC P12931 1/20 0.47
SLC2A1 P11166 1/20 0.47
ALDH1A1 P00352 3/20 0.44
KDM4E B2RXH2 2/20 0.44
HPGD P15428 2/20 0.44
HSD17B10 Q99714 1/20 0.44
PARP1 P09874 7/20 0.44
CHEK1 O14757 2/20 0.44
PIM1 P11309 2/20 0.44
AKT1 P31749 1/20 0.44
FLT3 P36888 1/20 0.44
PIM3 Q86V86 1/20 0.44
RPS6KA3 P51812 1/20 0.44
ALK Q9UM73 1/20 0.42
IP6K1 Q92551 3/20 0.42
IP6K3 Q96PC2 1/20 0.42
IP6K2 Q9UHH9 1/20 0.42
LCK P06239 1/20 0.41
FYN P06241 1/20 0.41
MKNK1 Q9BUB5 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8917 0.83 SRC (0.63) SRCSLC2A1ALDH1A1KDM4EPARP1
SCHEMBL23959894 0.82 SRC (0.49) SRCSLC2A1ALDH1A1HPGDPARP1
Acetic Acid SCHEMBL28399538 0.82 SLC2A1 (0.49) SRCSLC2A1ALDH1A1PARP1CHEK1
SCHEMBL6253346 0.82 SRC (0.52) SRCSLC2A1ALDH1A1PARP1CHEK1
SCHEMBL5374095 0.81 QPCT (0.48) ALDH1A1KDM4EHPGDHSD17B10LCK
SCHEMBL22029115 0.81 CHEK1 (0.51) SRCSLC2A1ALDH1A1PARP1CHEK1
SCHEMBL30591004 0.81 CHEK1 (0.51) SRCSLC2A1ALDH1A1PARP1CHEK1
SCHEMBL4141791 0.81 IP6K1 (0.52) SLC2A1ALDH1A1PARP1CHEK1PIM1
SCHEMBL298221 0.81 PARP1 (0.51) SRCSLC2A1ALDH1A1PARP1CHEK1
SCHEMBL4141934 0.81 SLC2A1 (0.54) SLC2A1ALDH1A1PARP1CHEK1PIM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090181958-A1 SUBSTITUTED NITROGEN-CONTAINING HETEROBICYCLES, THE PREPARATION THEREOF AND THEIR USE AS PHARMACEUTICAL COMPOSITIONS BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG (DE) 2009-07-16 US disclosed
US-7429597-B2 Substituted nitrogen-containing heterobicycles, the preparation thereof and their use as pharmaceutical compositions BOEHRINGER INGELHEIM PHARMA GMBH & CO., KG (DE) 2008-09-30 US disclosed
US-20040176603-A1 Substituted nitrogen-containing heterobicycles, the preparation thereof and their use as pharmaceutical compositions BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG (DE) 2004-09-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040176603-A1 Substituted nitrogen-containing heterobicycles, the preparation thereof and their use as pharmaceutical compositions F11, F12, F2 SRC 3074/4885SLC2A1 3168/4885ALDH1A1 2355/4885
US-20090181958-A1 SUBSTITUTED NITROGEN-CONTAINING HETEROBICYCLES, THE PREPARATION THEREOF AND THEIR USE AS PHARMACEUTICAL COMPOSITIONS F12, F11, F2 SRC 3097/4885SLC2A1 3473/4885ALDH1A1 3364/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.